Abstract
The synthesis of hetaryl 1,2,4-thiadiazolyl sulfides has been carried out by nucleophilic substitution of the chlorine atom in 5-chloro-1,2,3-thiadiazole by mercaptoheterocycles.
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REFERENCES
Al. Gommaa andM. Selhdar, Alexandria J. Pharm. Sci., 5, 153 (1991).
E. W. Tomas, Comprehensive Heterocyclic Chemistry, 2, Ed. by A. R. Katritzky,C. W. Rees, andE. F. Scriven, 4, 289 (1996).
E. G. Lebel,J. A. Ryals,L. Tharne,S. J. Uknes, andE. R. Ward, US Pat W098 03536; Chem. Abstr., 128, 137192 (1998).
F. Halgand,F. Vives.J.-P. Dumas,R. Cantegril,J. Gagnon,R. Douce,E. Forest, andD. Job, Biochemistry, 34, 4773 (1998).
L. C. Blaszczak,C. N. Eid,J. Flokowitsch,G. S. Gregory,S. A. Hitchock,G. W. Huffman,D. R. Mayhuhg,M. J. Nesler,D. A, Preston, andM. Zia-Ebrahimi, Bioorg. Med. Chem. Lett., 7, 2261 (1997).
T. Kobori,T. Hirada,M. Fujita,S. Kondo,T. Asada,S. Ono, andH. Tsuboi, Jpn. Pat. 09249665; Chem. Abstr., 127, 278196 (1998).
Yu. Yu. Morzherin,V. A. Bakulev,E. F. Dankova, andV. S. Mokrushin, Khim. Geterotsikl. Soedin., 548 (1994).
E. V. Tarasov,Yu. Yu. Morzherin,N. N. Volkova, andV. A. Bakulev, Khim. Geterotsikl. Soedin., 1124 (1996).
V. A. Bakulev,E. V. Tarasov,Yu. Yu. Morzherin.S. Toppet, andW. Dehaen, Bull. Soc. Chim. Belg., 106, 643 (1997).
E. V. Tarasov,Yu. Yu. Morzherin,S. Toppet,W. Dehaen, andV. A. Bakulev, J. Chem. Res., 11, (S) 396, (M) 2472 (1997).
V. A. Bakulev,E. V. Tarasov,Yu. Yu. Morzherin,I. Lutyen,S. Toppet, andW. Dehaen, Tetrahedron, 54, 8501 (1998).
G. L'abbe,P. Delbeke,L. Bastin,W. Dehaen, andS. Toppet, J. Heterocycl. Chem., 30, 301 (1993).
M. J. S. Dewar andE. G. Zoebisch, Theochem., 49, 1 (1988).
V. S. Mokrushin, Diss. Dr. Sc. (Chem.), Moscow (1985).
J. Goerdeler andG. Gnad, Chem. Ber., 99, 1618 (1966).
Yu. Yu. Morzherin,E. V. Tarasov, andV. A. Bakulev, Khim. Geterotsikl. Soedin., 554 (1994).
V. A. Bakulev, Diss. Dr. Sc. (Chem.), Moscow (1990).
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Morzherin, Y.Y., Pospelova, T.A., Glukhareva, T.V. et al. Hetaryl 1,2,3-Thiadiazolyl Sulfides. Chemistry of Heterocyclic Compounds 37, 1270–1278 (2001). https://doi.org/10.1023/A:1013861930028
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DOI: https://doi.org/10.1023/A:1013861930028