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Chemistry of Heterocyclic Compounds

, Volume 48, Issue 2, pp 355–357 | Cite as

Copper-catalyzed arylation of tetrazole-5-thiones upon convection heating and microwave activation conditions

  • U. N. Dmitrieva
  • S. M. Ramsh
  • Yu. E. Zevatskii
  • T. V. Artamonova
  • L. V. MyznikovEmail author
Article

The arylation of 1-phenyltetrazole-5-thione using a series of iodobenzene derivatives in the presence of cuprous chloride and a ligand such as ethylenediamine. It was shown that the use of microwave activation permitted shortening of the reaction time, increasing yields and simplification of the reaction products isolation.

Keywords

aryl iodide cuprous chloride ethylenediamine tetrazole-5-thione arylation microwave activation 

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Copyright information

© Springer Science+Business Media, Inc. 2012

Authors and Affiliations

  • U. N. Dmitrieva
    • 1
  • S. M. Ramsh
    • 1
  • Yu. E. Zevatskii
    • 1
  • T. V. Artamonova
    • 1
  • L. V. Myznikov
    • 1
    Email author
  1. 1.St. Petersburg State Technological Institute (Technical University)Saint PetersburgRussia

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