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Synthesis of 2-hetaryl-3-(indol-1-yl)-and -(3-pyrrol-1-yl)maleimides and study of their conversions under the action of protic acids*

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Chemistry of Heterocyclic Compounds Aims and scope

A series of 3-(indol-1-yl)maleimides has been synthesized, substituted at position 2 by residues of amines or various nitrogenous heterocycles. The possibility of obtaining new polycondensed heterocyclic structures from them has been studied. Experimental investigations confirmed theoretical predictions made on the basis of results of quantum-chemical calculations.

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Authors and Affiliations

  1. G. F. Gause Institute of New Antibiotics, Russian Academy of Medical Sciences, Moscow, 119021, Russia

    S. A. Lakatosh, E. E. Bykov & M. N. Preobrazhenskaya

Authors
  1. S. A. Lakatosh
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  2. E. E. Bykov
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  3. M. N. Preobrazhenskaya
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Corresponding author

Correspondence to S. A. Lakatosh.

Additional information

*Dedicated to the shining memory of A. N. Kost.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 10, pp. 1515-1525, October, 2010.

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Lakatosh, S.A., Bykov, E.E. & Preobrazhenskaya, M.N. Synthesis of 2-hetaryl-3-(indol-1-yl)-and -(3-pyrrol-1-yl)maleimides and study of their conversions under the action of protic acids*. Chem Heterocycl Comp 46, 1224–1232 (2011). https://doi.org/10.1007/s10593-011-0656-9

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  • DOI: https://doi.org/10.1007/s10593-011-0656-9

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