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Synthesis and reactions of thioamides of 5-amino-2-aryl-2H-1,2,3-triazole-4-carboxylic acid

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Chemistry of Heterocyclic Compounds Aims and scope

A method has been developed for obtaining thioamides of 5-amino-2-aryl-2H-1,2,3-triazole-4-carboxylic acid. Their heterocyclization reactions with bifunctional reagents has been studied. New heterocyclic polycyclic ensembles have been synthesized containing a 1,2,3-triazole fragment, a thiazole, and a residue of the natural alkaloid cytisine.

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Correspondence to N. P. Belskaya.

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Dedicated to Academician of the Russian Academy of Sciences O. N. Chupakhin on his 75th jubilee.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 7, pp. 1061–1071, July, 2009.

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Belskaya, N.P., Sapozhnikova, S.G., Bakulev, V.A. et al. Synthesis and reactions of thioamides of 5-amino-2-aryl-2H-1,2,3-triazole-4-carboxylic acid. Chem Heterocycl Comp 45, 844–852 (2009). https://doi.org/10.1007/s10593-009-0348-x

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  • DOI: https://doi.org/10.1007/s10593-009-0348-x

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