Abstract
It has been established that the interaction of N1-(2-hydroxyphenylmethylthieno[2,3-b]pyrid-3-yl)arylamides with hydrazine hydrate leads to thieno[2,3-b]pyridine-2,3-diamines. It was shown that the reaction of the latter with acetylacetone and acetoacetic ester occurs regioselectively at the amino group in position 3 of the thiophene ring.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, pp. 1400–1408, September, 2007.
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Lipunov, M.M., Kaigorodova, E.A., Konyushkin, L.D. et al. Synthesis and reactivity of thieno[2,3-b]pyridine-2,3-diamines. Chem Heterocycl Comp 43, 1189–1196 (2007). https://doi.org/10.1007/s10593-007-0182-y
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DOI: https://doi.org/10.1007/s10593-007-0182-y