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Synthesis of novel 5-piperidyl-substituted 7-hydroxy-3H-1,2,3-triazolo[4,5-d]pyrimidines

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

A series of 8-azapurin-6-ones having a piperidine substituent at position 5 has been synthesized from pipecolinate esters, benzylazides, and cyanoacetamide.

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Authors and Affiliations

  1. D. I. Mendeleev Russian University of Chemical Technology, Moscow, 125047, Russia

    K. V. Kuleshov, K. Yu. Borovkov, O. G. Rodin & V. P. Perevalov

Authors
  1. K. V. Kuleshov
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  2. K. Yu. Borovkov
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  3. O. G. Rodin
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  4. V. P. Perevalov
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 2, pp. 276–290, February, 2006.

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Kuleshov, K.V., Borovkov, K.Y., Rodin, O.G. et al. Synthesis of novel 5-piperidyl-substituted 7-hydroxy-3H-1,2,3-triazolo[4,5-d]pyrimidines. Chem Heterocycl Compd 42, 246–260 (2006). https://doi.org/10.1007/s10593-006-0078-2

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  • DOI: https://doi.org/10.1007/s10593-006-0078-2

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