Abstract
By recyclization of 2-R-6-ethyl-7-hydroxy(methoxy)-3-(5-phenyl-1,3,4-thiadiazol-2-yl)chromones when treated with hydrazine hydrate and phenylhydrazine, we synthesized 5-phenyl-2-(3-R-5-R1-1H-pyrazol-4-yl)-1H-1,3,4-thiadiazoles and 2-(3-R-5-R1-1-phenyl-1H-pyrazol-4-yl)-5-phenyl-1H-1,3,4-thiadiazoles. We confirmed the structure of the latter from 1H NMR spectra.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 5, pp. 781–787, May, 2005.
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Shokol, T.V., Semenyuchenko, V.V. & Khilya, V.P. 5-Phenyl-2-(pyrazol-4-yl)-1,3,4-thiadiazoles. Chem Heterocycl Compd 41, 673–678 (2005). https://doi.org/10.1007/s10593-005-0201-9
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DOI: https://doi.org/10.1007/s10593-005-0201-9