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Facile synthesis and biological evaluation of heterocyclic compounds containing Diazepam

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  • Medicinal Chemistry & Natural Products
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Abstract

Diazepamoxadiazoles4,5,6,12,14 and22 were prepared with the binary form system. Diazepamthiadiazoles15,20 and Diazepamtriazoles7,8,9,17,18,19 and21 were also shapely synthesized. Some of these compounds were screened to test their antibacterial activity againstE. coli andB. subtilis compounds 15 and 20 show potent activity against these bacteria.

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  1. Department of Chemistry, Faculty of Science, Mansoura University, Mansoura, Egypt

    M. A. Berghot

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  1. M. A. Berghot
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Correspondence to M. A. Berghot.

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Berghot, M.A. Facile synthesis and biological evaluation of heterocyclic compounds containing Diazepam. Arch Pharm Res 24, 263–269 (2001). https://doi.org/10.1007/BF02975089

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  • DOI: https://doi.org/10.1007/BF02975089

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