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Chemistry of Heterocyclic Compounds

, Volume 33, Issue 5, pp 600–604 | Cite as

4-Hydroxy-2-quinolones. 32. Synthesis and antithyroid activity of thio analogs of 1H-2-oxo-3-(2-Benzimidazolyl)-4-hydroxyquinoline

  • I. V. Ukrainets
  • S. G. Taran
  • O. V. Gorokhova
  • N. A. Marusenko
  • A. V. Turov
Article

Abstract

We propose preparative synthesis methods for 2-thio-4-hydroxy-, 2-oxo-4-mercapto-, and 2-thio-4-mercapto-1H-3-(2-benzimidazolyl)quinolines. We have studied the antithyroid activity of the synthesized compounds.

Keywords

Organic Chemistry Quinoline Synthesis Method Thio Hydroxyquinoline 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Plenum Publishing Corporation 1997

Authors and Affiliations

  • I. V. Ukrainets
  • S. G. Taran
  • O. V. Gorokhova
  • N. A. Marusenko
  • A. V. Turov

There are no affiliations available

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