Abstract
Treatment of 4-aryl-5-aminopyrazoles and 2-aryl-3-amino-maleimides with tris(morpholino)methane gives N-azolyl formamidines which are converted upon heating in trifluoroacetic acid to polycondensed heterocycles with isoquinoline and indolo[2,3-c]pyridine structural fragments.
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L. M. Litvinenko Institute of Physico-Organic and Carbon Chemistry, Ukrainian Academy of Sciences, Donetsk 340114. A. N. Kosygin State Textile Academy, Moscow 117918 GSP-1. Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 1, pp. 80–84, January, 1997.
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Bogza, S.D., Ivanov, A.V., Dulenko, V.I. et al. Cyclodesamination of N-azolylformamidines. Synthesis of polyazaheterocycles with isoquinoline and indolo[2,3-c]-pyridine structural fragments. Chem Heterocycl Compd 33, 69–73 (1997). https://doi.org/10.1007/BF02290749
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DOI: https://doi.org/10.1007/BF02290749