Abstract
A new method is proposed for the synthesis of substitituted 2,5-diazabicyclo[2.2.1]heptanes from 1-(tert-butoxycarbonyl)-4-tosyloxy-2-(tosyloxymethyl)pyrrolidine.1H NMR spectroscopy indicated multiple conformations of 2-(tert-butoxycarbonyl)-2,5-diazabicyclo[2.2.1]heptanes in solution.
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St. Petersburg State University, 198904 St. Petersburg, Russia. Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 4, pp. 501–503, April, 2000.
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Yakovlev, M.E., Lobanov, P.S. & Potekhin, A.A. Synthesis of substituted 2,5-diazabicyclo[2.2.1]heptanes. Chem Heterocycl Compd 36, 429–431 (2000). https://doi.org/10.1007/BF02269540
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DOI: https://doi.org/10.1007/BF02269540