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Acylation of 2- and 4-hydroxyaminopyrimidines

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Monoacylation of alkyl (aryl)-containing 2- and 4-hydroxyaminopyrimidines with acid anhydrides and acid chlorides leads preferentially to the acyloxyamino-pyrimidines; the corresponding reaction with isocyanates leads to the (N-car-bamoyl)hydroxyaminopyrimidines.

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Deceased.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 5, pp. 654–658, May, 1988.

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Sedova, V.F., Moskalenko, G.G. & Mamaev, V.P. Acylation of 2- and 4-hydroxyaminopyrimidines. Chem Heterocycl Compd 24, 533–537 (1988). https://doi.org/10.1007/BF00755695

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  • DOI: https://doi.org/10.1007/BF00755695

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