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Synthesis, stereochemistry, and isomeric transformations of 4-aryl-5-aroyl-2-methylthio-2-imidazolines

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Abstract

The corresponding 4-aryl-5-aroyl-2-methylthio-2-imidazolines were obtained by the reaction of complexes of cis- and trans-3-aroylaziridines and boron trifluoride with methyl thiocyanate. It is shown on the basis of spectral data that the aziridine ring is opened regiospecifically at the C(2) atom and stereospecifically with inversion of the configuration.

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Authors and Affiliations

  1. A. N. Sevchenko Scientific-Research Institute of Applied Physical Problems, 220065, Minsk

    V. A. Konovalov, O. N. Bubel' & I. G. Tishchenko

Authors
  1. V. A. Konovalov
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  2. O. N. Bubel'
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  3. I. G. Tishchenko
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Additional information

Deceased.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1484–1488, November, 1988.

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Konovalov, V.A., Bubel', O.N. & Tishchenko, I.G. Synthesis, stereochemistry, and isomeric transformations of 4-aryl-5-aroyl-2-methylthio-2-imidazolines. Chem Heterocycl Compd 24, 1229–1233 (1988). https://doi.org/10.1007/BF00633501

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  • DOI: https://doi.org/10.1007/BF00633501

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