Abstract
N-Alkylaminothiophene derivatives were obtained by the reaction of 3-hydroxy-4-carbethoxy-5-methylthiophene with alkylammonium acetates, while N-arylaminothiophene derivatives were obtained by the reaction of the same thiophene derivative with aromatic amines in the presence of catalytic amounts of iodine.
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Translated from Khimiya Geterotsilicheskikh Soedinenii, No. 12, pp. 1602–1604, December, 1970.
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Shvedov, V.I., Vasil'eva, V.K. & Grinev, A.N. Alkyl- and arylamination of 3-hydroxy-4-carbethoxy-5-methylthiophene. Chem Heterocycl Compd 6, 1495–1497 (1970). https://doi.org/10.1007/BF00522564
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DOI: https://doi.org/10.1007/BF00522564