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Electrophilic substitution reactions of acylated 2-aminoindole derivatives

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

The bromination, nitration, and acylation reactions of various acyl derivatives belonging to the 2-aminoindole series of compounds have been investigated. It has been found that substitution occurs both at the β-carbon atom as well as at the 5- and 6-positions of the benzene ring. The ratio of reaction products depends upon the nature of the electrophile as well as on the degree of substitution of the 2-aminoindole.

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Authors and Affiliations

  1. M. V. Lomonosov Moscow State University, Moscow

    E. S. Besidskii, G. A. Golubeva & L. A. Sviridova

Authors
  1. E. S. Besidskii
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  2. G. A. Golubeva
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  3. L. A. Sviridova
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 7, pp. 941–945, July, 1985.

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Besidskii, E.S., Golubeva, G.A. & Sviridova, L.A. Electrophilic substitution reactions of acylated 2-aminoindole derivatives. Chem Heterocycl Compd 21, 782–785 (1985). https://doi.org/10.1007/BF00519147

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  • DOI: https://doi.org/10.1007/BF00519147

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