Abstract
The reaction of methyl aziridine-2-carboxylate with hydrazine or alkylhydrazines gives the respective hydrazides, which with ketones form 2,2-disubstituted 1,3,4-triazabicyclo-[4.1.0] heptan-5-ones. With aldehydes they form the respective hydrazones. The reaction of the amide and methyl ester of aziridine-2-carboxylic acid with aldehydes gives a series of aziridinocarbinols.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 6, pp. 774–778, June, 1985.
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Trapentsier, P.T., Kalvin'sh, I.Y., Liepin'sh, É.É. et al. Reactions of aziridine-2-carboxylic acid derivatives with aldehydes and ketones. Chem Heterocycl Compd 21, 646–650 (1985). https://doi.org/10.1007/BF00515064
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DOI: https://doi.org/10.1007/BF00515064