Abstract
Acetylenic α-aziridinocarbinols were obtained by reaction of propiolaldehyde and phenylpropiolaldehyde with aziridine and its 2-substituted derivatives. The mechanism of the conversion of the latter to β-aziridinoacroleins was studied.
Article PDF
Similar content being viewed by others
Literature cited
R. G. Kostyanovskii, Dokl. Akad. Nauk SSSR, 135, 8531 (1960).
T. Maruyma, N. Kuroki, and K. Konishi, Bull. Univ. Osaka Prefast., A13, 135 (1964).
K. Tsou, K. Hoegerle, and H. Su, J. Med. Chem., 6, 435 (1963).
R. G. Kostyanovskii and V. F. Bystrov, Izv. Akad. Nauk SSSR, Otd. Khim. Nauk, 1448 (1962).
R. G. Kostyanovskii and V. F. Bystrov, Izv. Akad. Nauk SSSR, Otd. Khim. Nauk, 171 (1963).
S. A. Giller and M. Yu. Lidak, Methods for the Synthesis of and Investigation of Antitumorigenic Preparations [in Russian], Medgiz, Moscow (1962), p. 193.
M. Yu. Lidak and S. A. Giller, Izv. Akad. Nauk LatvSSR, Ser. Khim., No. 1, 81 (1961).
R. G. Kostyanovskii, O. Ya. Pan'shin, and G. Z. Papoyan, Dokl. Akad. Nauk SSSR, 177, 1099 (1967).
H. Betian, Ann., 566, 210 (1950).
A. Mannshreck, R. Radeglia, E. Grundemann, and R. Ohme, Chem. Ber., 100, 1778 (1967).
J. M. Lehn, Fortschr. Chem. Forsch., 15, 311 (1970).
Author information
Authors and Affiliations
Additional information
Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 2, pp. 207–212, February, 1977.
Rights and permissions
About this article
Cite this article
Eremeev, A.V., Tikhomirov, D.A. & Liepin'sh, É.É. Acetylenicα-aziridinocarbinols and the mechanism of their conversion to β-aziridinoacroleins. Chem Heterocycl Compd 13, 165–170 (1977). https://doi.org/10.1007/BF00497869
Received:
Revised:
Issue Date:
DOI: https://doi.org/10.1007/BF00497869