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Selective alkylation of imidazole-4(5)-carboxamides

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Alkylation of imidazole-4(b)-carboxamides by alkyl halides or dimethylsulfate leads to the selective formation of 1-alkyl-imidazole-4-carboxamides.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 4, pp. 475–477, April, 1990.

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Piotrovskii, L.B., Dumpis, M.A. Selective alkylation of imidazole-4(5)-carboxamides. Chem Heterocycl Compd 26, 407–409 (1990). https://doi.org/10.1007/BF00497210

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  • DOI: https://doi.org/10.1007/BF00497210

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