Chemistry of Heterocyclic Compounds

, Volume 26, Issue 5, pp 520–524 | Cite as

Rearrangement of 1-acetylindoxyl oxime to 1-acetyl-2-chloro-3-iminoindoline hydrochloride

  • V. S. Velezheva
  • S. Yu. Ryabova


Rearrangement of 1-acetylindoxyl oxime upon treatment with hydrogen chloride in acetic acid results in the formation of 1-acetyl-2-chloro-3-iminoindoline hydrochloride. Hydrolysis and acylation of the latter have been studied, along with reaction of 1-acetyl-2-chloro-3-(Ω-chloroacetyl)aminoindole with N- and S-nucleophiles.


Hydrogen Acetic Chloride Hydrolysis Acetic Acid 
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Literature Cited

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Copyright information

© Plenum Publishing Corporation 1990

Authors and Affiliations

  • V. S. Velezheva
    • 1
  • S. Yu. Ryabova
    • 1
  1. 1.S. Ordzhonikidze All-Union Scientific Research Chemical Pharmaceutical InstituteMoscow

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