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Indole chemistry

XXVII. 2-Haloacetylindoles

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

A number of 2-haloacetylindoles were synthesized from substituted 2-diazoacetylindoles. The direct bromination of 3-methyl-2-acetylindole proceeds at the acetyl group of form 3-methyl-2-bromaoacetylindole. In 2-acetylindole, the CH3 group and the 3-position of the pyrrole ring are simultaneously brominated.

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Literature cited

  1. L. G. Yudin, A. N. Kost, and A. I. Pavlyuchenko, Khim. Geterotsikl. Soedin., 1517 (1971).

  2. K. Bodendorf and A. Walk, Arch. Pharm., 294, 484 (1961).

    Google Scholar 

  3. S. S. Liberman, G. P. Sukhinina, L. M. Orlova, M. N. Preobrazhenskaya, Z. G. Starostina, and N. N. Suvorov, Khim.-Farmats. Zh., No. 3, 22 (1969).

    Google Scholar 

  4. T. Nogrady, T. Doyle, and L. Morris, J. Med. Chem., 8, 656 (1965).

    Google Scholar 

  5. Q. Mingoia, Gazz. Chim. Ital., 61, 646 (1931).

    Google Scholar 

  6. D. Ames, R. Bowman, D. Evans, and W. Jones, J. Chem. Soc., 1984 (1956).

  7. R. Sundberg, J. Org. Chem., 30, 3604 (1965).

    Google Scholar 

  8. J. De Graw, J. Kennedy, and W. Skinner, J. Heterocycl. Chem., 3, 9 (1966).

    Google Scholar 

  9. M. N. Preobrazhenskaya, L. M. Orlova, and N. N. Suvorov, Zh. Vsesoyuzn. Khim. Obshchesta, 13, 236 (1968).

    Google Scholar 

  10. A. J. Namis, E. Cortés, O. Collera, and F. Walls, Boletin Instituto Quimico, Univ. Nacional México, 18, 64 (1966).

    Google Scholar 

  11. M. Matell, Arkiv Kemi, 10, 179 (1956).

    Google Scholar 

  12. L. Bellamy, Infrared Spectra of Complex Molecules, Methuen (1958).

  13. A. N. Kost, R. S. Sagitullin, V. I. Gorbunov, and G. I. Barinova, Khim.-Farmats. Zh., No. 3, 14 (1967).

    Google Scholar 

  14. K. Ishizumi, T. Shiori, and S. Jamade, Chem. Pharm. Bull. (Tokyo), 15, 863 (1967); Chem. Abstr., 67, 108,510 (1967).

    Google Scholar 

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Authors and Affiliations

  1. Novokuznetsk Scientific-Research Institute of Pharmaceutical Chemistry, M. V. Lomonosov Moscow State University, USSR

    A. N. Kost, S. M. Gorbunova & V. A. Budylin

Authors
  1. A. N. Kost
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  2. S. M. Gorbunova
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  3. V. A. Budylin
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Additional information

See [1] for communication XXVI.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1522–1526, November, 1971.

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Kost, A.N., Gorbunova, S.M. & Budylin, V.A. Indole chemistry. Chem Heterocycl Compd 7, 1416–1420 (1971). https://doi.org/10.1007/BF00481108

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  • DOI: https://doi.org/10.1007/BF00481108

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