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Chemistry of Heterocyclic Compounds

, Volume 13, Issue 10, pp 1122–1126 | Cite as

Synthesis of derivatives of pyrido[3,4-b]- and azepino[3,4-b]pyrrolo[2,3-d]pyrimidines from enamines of α-oxo lactams

  • R. G. Glushkov
  • I. M. Zasosova
  • I. M. Ovcharova
Article
  • 23 Downloads

Abstract

The reaction of enamines of some α-oxo lactams with 1,3-dimethyl- and 1,3-dibenzyl-4-hydrazinouracils gave the uracilyl-4-hydrazones of these lactams, the catalytic and thermal indolization of which yielded derivatives of pyrido[3,4-b]- and azepino[3,4-b]pyrrolo[2,3-d]pyrimidines. Some reactions of the latter were studied.

Keywords

Organic Chemistry Pyrimidine Lactam Enamine 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Plenum Publishing Corporation 1978

Authors and Affiliations

  • R. G. Glushkov
    • 1
  • I. M. Zasosova
    • 1
  • I. M. Ovcharova
    • 1
  1. 1.S. Ordzhonikidze All-Union Scientific-Research Pharmaceutical-Chemistry InstituteMoscow

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