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Synthesis of 2-cyclohexylcarbonyl-4-oxoperhydropyrazino [2,1-a]-isoquinoline

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

2-Cyclohexylcarbonyl-4-oxoperhydropyrazino [2,1-alisoquinoline, an analog of the highly effective anthelmintic prasiquantel, was synthesized from 2-(cyclohexen-1-yl)-ethylamine.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 8, pp. 1115–1118, August, 1988.

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Tsizin, Y.S., Sergovskaya, N.L. & Shekhter, O.V. Synthesis of 2-cyclohexylcarbonyl-4-oxoperhydropyrazino [2,1-a]-isoquinoline. Chem Heterocycl Compd 24, 920–922 (1988). https://doi.org/10.1007/BF00479350

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  • DOI: https://doi.org/10.1007/BF00479350

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