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Indole chemistry

XXVIII. 2-oxo-α-carbolines

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

The condensation of 1-substituted 2-aminoindoles with β-keto esters gives 2-oxo-α-carbolines. Substitution of diketenes for the β-keto esters leads to a mixture of 2-oxo- and 4-oxo- compounds.

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See [1] for communication XXVII.

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 1, pp. 48–54, January, 1972.

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Borisov, N.N., Sagitullin, R.S. & Kost, A.N. Indole chemistry. Chem Heterocycl Compd 8, 46–51 (1972). https://doi.org/10.1007/BF00478490

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  • DOI: https://doi.org/10.1007/BF00478490

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