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Synthesis of 2, 6-diamino-8-arylpurines using aromatic aldehydes

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

2,6-Diamino-8-arylpurines were obtained by condensation of 2,4,5,6-tetraaminopyrimidine with aromatic aldehydes with nitrobenzene as the oxidizing agent in the presence of p-toluenesulfonic acid or divalent copper.

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Authors and Affiliations

  1. N. N. Petrov Scientific-Research Institute of Oncology, Ministry of Health of the USSR, Leningrad

    V. S. Kuznetsov & A. L. Remizov

Authors
  1. V. S. Kuznetsov
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  2. A. L. Remizov
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 10, pp. 1430–1434, October, 1972.

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Kuznetsov, V.S., Remizov, A.L. Synthesis of 2, 6-diamino-8-arylpurines using aromatic aldehydes. Chem Heterocycl Compd 8, 1292–1297 (1972). https://doi.org/10.1007/BF00475551

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  • DOI: https://doi.org/10.1007/BF00475551

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