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Synthesis of 1-(arylethynyl)aziridines

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Studies have been made on the possible synthesis of 1-(arylethynyl)aziridines by oxidative condensation of phenylacetylene with aziridine and by alkylation of aziridine with 1-halo-2-arylacetylenes.

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Literature Cited

  1. D. A. Tikhomirov, Yu. V. Shubina, and A. V. Eremeev, Khim. Geterotsikl. Soedin., No. 11, 1492 (1984).

    Google Scholar 

  2. Yu. V. Shubina, D. A. Tikhomirov, and A. V. Eremeev, Khim. Geterotsikl. Soedin., No. 5, 618 (1985).

    Google Scholar 

  3. L. I. Peterson, Tetrahedron Lett., No. 51, 5357 (1968).

    Google Scholar 

  4. R. Huisgen, B. Geise, and H. Huber, Tetrahedron Lett., No. 20, 1883 (1967).

    Google Scholar 

  5. V. Wolf and F. Kowitz, Ann. Chem., 638, 33 (1960).

    Google Scholar 

  6. S. I. Miller and J. I. Dickstein, Acc. Chem. Res., 9, 358 (1976).

    Google Scholar 

  7. V. Wolf and W. Block, Ann. Chem., 637, 119 (1960).

    Google Scholar 

  8. V. Wolf and H. Piater, Ann. Chem., 696, 90 (1966).

    Google Scholar 

  9. P. Beltrame, A. Gavezzoti, and M. Simonetta, J. Chem. Soc., Perkin Trans. 2, No. 3, 502 (1974).

    Google Scholar 

  10. E. F. V. Scriven, Chem. Soc. Rev., 12, 129 (1983).

    Google Scholar 

  11. H. J. Bestmann and H. Frey, Ann. Chem., No. 12, 2061 (1980).

    Google Scholar 

  12. M. Makosza and M. Fedorinski, Roczn. Chem., 49, 1779 (1975).

    Google Scholar 

  13. Dictionary of Organic Compounds, Vol. 5 (1982), p. 4590.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 1, pp. 39–43, January, 1987.

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Tikhomirov, D.A., Eremeev, A.V. Synthesis of 1-(arylethynyl)aziridines. Chem Heterocycl Compd 23, 30–34 (1987). https://doi.org/10.1007/BF00475469

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  • DOI: https://doi.org/10.1007/BF00475469

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