Abstract
A method has been proposed for the detosylation of 3-substituted pyrroles by potassium in tetrahydrofuran with a simultaneous activation of the 1-position for the subsequent alkylation or acylation of the pyrrolepotassium derivative.
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Translated from Khimiya Geterotsiklicheskih Soedinenii, No. 5 pp. 634–635, May, 1991,
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Vorob'eva, S.L., Magedov, I.V. & Traven', V.F. A convenient method of synthesis of 1,3-disubstituted pyrroles. Chem Heterocycl Compd 27, 504–505 (1991). https://doi.org/10.1007/BF00473993
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DOI: https://doi.org/10.1007/BF00473993