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In memory of Solomon Aronovich Giller

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Chemistry of Heterocyclic Compounds Aims and scope

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I. Chemistry of Furan

  1. S. A. Giller and A. A. Berzin', “Crystalline modifications of 5-nitro-2-furfurylidenea-inoguanidine sulfate,” Izv. Akad. Nauk LatvSSR, No. 11, 1733–1738 (1951).

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  2. S. A. Giller and Ya. A. Éidus, “UV absorption spectra of some nitrofurans,” Izv. Akad. Nauk LatvSSR, No. 8, 1223–1238 (1951).

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  3. S. A. Giller, “Study of methods for the synthesis and physicochemical properties of and interrelationship between the structure and biological activity of some substituted 5-trofurfurylideneimines,” Author's Abstract of His Master's Degree, Riga (1953).

  4. S. A. Giller, “Nitrofurans,” in: Furacilin and Experience with Its Application [in Russian], Riga (1953), pp. 7–74.

  5. S. A. Giller and A. A. Berzin', “Crystalline modifications of 5-nitro-2-furfurylidenea-minoguanidine sulfate,” in: Furacilin and Experiences with Its Application [in Russian], Riga (1953), pp. 91–96.

  6. S. A. Giller, N. O. Saldabol, and Ya. A. Éidus, “Some studies of the UV absorption spectra of nitrofurans,” Izv. Akad. Nauk SSSR, Ser. Fiz., 708–714 (1953).

  7. S. A. Giller and Ya. A. Éidus,* “UV absorption spectra of some nitrofurans,” in: Furacilin and Experience with Its Application [in Russian], Riga (1953), pp. 75–90.

  8. S. A. Giller, M. M. Gershov, N. N. Naumenko, and É. Yu. Gudrinietse, “Method for the preparation of 5-nitrofurfural diacetate,” USSR Author's Certificate No. 97012; Byul. Izobr., No. 2, 14 (1954).

  9. S. A. Giller and M. Ya. Berklava, “Acetylation in the presence of anhydrous zinc chloride,” Izv. Akad. Nauk LatvSSR, No. 4, 53–59 (1956).

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  10. S. A. Giller, “Nitrofurans,” in: Problems in the Utilization of Pentosan-Containing Raw Material. Proceedings of the All-Union Conference [in Russian], Riga (1958), pp. 451–458.

  11. S. A. Giller, A. É. Berzinya, and L. Ya. Lauberte, “Research on the alkylation of furan with olefins. I. Alkylation of furan with ethylene,” Izv. Akad. Nauk LatvSSR, No. 4, pp. 71–79 (1958).

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  12. S. A. Giller and K. K. Venter, “Syntheses involving 5-nitrofuryl-2-polyalkenals and 5-nitrofuryl-2-polyalkenones. I. Preparation of β-(5-nitro-2-furyl) acrolein by condensation of 5-nitrofurfural with acetaldehyde,” Izv. Akad. Nauk LatvSSR, No. 12, pp. 115–124 (1958).

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  13. S. A. Giller and Z. Ya. Zelmene, “Some new furan mercurichlorides,” Izv. Akad. Nauk LatvSSR, No. 11, pp. 97–101 (1958).

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  14. S. A. Giller and G. P. Sokolov, “Multiplicity of.the bond between the 3 and 4 atoms in the furan ring,” Izv. Akad. Nauk LatvSSR, No. 12, 125–128 (1958).

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  15. N. O. Saldabol and S. A. Giller, “Syntheses in the 2-acetylfuran series,” in: Problems in the Utilization of Pentosan-Containing Raw Material. Proceedings of the All-Union Conference [in Russian], Riga (1958), pp. 379–391.

  16. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. I. Nitration of methyl 2-furyl ketone,” Izv. Akad. Nauk LatvSSR, No. 10, 101–108 (1958).

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  17. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. II. ω-Bromination of methyl 2-furyl ketone and its 5-nitro derivative,” Izv. Akad. Nauk LatvSSR, No. 11, 91–96 (1958).

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  18. K. K. Venter, S. A. Giller, and N. O. Saldabol, “Syntheses involving 5-nitrofuryl-2-polyalkenals and 5-nitrofuryl-2-polyalkenones. II. Nitration of 2-furfurylideneacetone,” Izv. Akad. Nauk LatvSSR, No. 8, 99–106 (1959).

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  19. S. A. Giller and A. É. Berzinya, “Research on the alkylation of furan with olefins. II. Magnitude of the increment of the molecular refractions of mono- and polyalkylfurans,” Izv. Akad. Nauk LatvSSR, No. 5, 109–114 (1959).

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  20. S. A. Giller and M. Ya. Berklava, “Some comments on the nitration of 2-furyl-β-nitroethylene,” Izv. Akad. Nauk LatvSSR, 115–119 (1959).

  21. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. III. Aminomethyl 2-furyl ketone and some of its derivatives,” Izv. Akad. Nauk LatvSSR, No. 1, 77–85 (1959).

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  22. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. IV. ω-Dialkylsulfonium derivatives of methyl 2-furyl ketone and methyl 5-nitro-2-furyl ketone,” Izv. Akad. Nauk LatvSSR, No. 3, 53–56 (1959).

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  23. S. A. Giller, B. V. Kurgan, and N. O. Saldabol, “Preparative method for the synthesis of 5-nitropyromucic acid,” Izv. Akad. Nauk LatvSSR, No. 3, 49–51 (1959).

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  24. S. A. Giller and G. P. Sokolov, “Tetrahydrofuran as a solvent for the reduction of carbonyl-containing compounds,” Izv. Akad. Nauk LatvSSR, No. 2, 85–90 (1959).

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  25. N. O. Saldabol, B. V. Kurgan, and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. V. Hydroxymethyl 2-furyl ketone and some of its derivatives,” Izv. Akad. Nauk LatvSSR, No. 4, 81–86 (1959).

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  26. S. A. Giller, K. K. Venter, N. O. Saldabol, and R. Yu. Kalnberg, “Method for the preparation of β-(5-nitro-2-furyl) acrolein and α-ethyl-β-(5-nitro-2-furyl) acrolein,” USSR Author's Certificate No. 130045; Byul. Izobr., No. 14, 15 (1960).

  27. É. Ya. Lukevits, Yu. P. Romadan, and S. A. Giller, “Synthesis of furfuryloxysilanes,” Izv. Akad. Nauk LatvSSR, No. 7, 59–64 (1961).

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  28. K. K. Venter, S. A. Giller, and A. A. Lazdyn'sh, “Syntheses involving 5-nitrofuryl-2-polyalkenals and 5-nitrofuryl-2-polyalkenones. IV. Nitration of β-(2-furyl) acrolein and synthesis of some unsaturated furan aldehydes and ketones,” Izv. Akad. Nauk LatvSSR, No. 5, 87–97 (1961).

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  29. N. O. Saldabol and S. A. Giller, “New Mannich bases from 2-acetylfuran, 2-furalacetone, and their 5-nitro derivatives,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 309–310 (1962).

  30. K. K. Venter, S. A. Giller, and V. V. Tsirule, “Nitration of β- (5-nitro-2-furyl) acrylic acid derivatives,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 131–134 (1962).

  31. S. A. Giller and A. É. Berzinya, “Research on the alkylation of furan with olefins. III. Alkylation of furan with propylene,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 103–111 (1962).

  32. S. A. Giller and A. É. Berzinya, “Research on the alkylation of furan with olefins. IV. Alkylation of furan with 1-butene and isobutylene,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 113–118 (1962).

  33. S. A. Giller and A. É. Berzinya, “Research on the alkylation of furan with olefins. V. Alkylation of furan with isoamylenes,” Izv. Akad. Nauk, SSR, Ser. Khim., 445–453 (1962).

  34. É. Ya. Lukevits, Yu. P. Romadan, S. A. Giller, and M. G. Voronkov, “Organosilicon compounds of the furan series. Syntheses in a series of furan-containing organosilicon compounds. III. Organosilicon derivatives of furylcarbinols and 5-substituted furfuryl alcohols,” Dokl. Akad. Nauk SSSR, 14, 806–808 (1962).

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  35. G. P. Sokolov and S. A. Giller, “Method for the preparation of 2,2,5-trimethoxy-2,5,-dihydrofuran,” USSR Author's certificate No. 149430; Byul. Izobr., No. 16, 25 (1962).

  36. M. Ya. Berklava and S. A. Giller, “Alcohols of the nitrofuran series. I. Reduction of 5-nitrofurfural and β-(5-nitro-2-furyl) acrolein with sodium borohydride and esterification of the resulting alcohols,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 349–355 (1963).

  37. S. A. Giller, N. O. Saldabol, and A. Ya. Medne, “2-Amino-4-(5-nitro-2-furyl) thiazole and its derivatives,” Zh. Obshch. Khim., 33, 317–318 (1963).

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  38. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. VI. New ω-ammonium derivatives of methyl 2-furyl ketone. Utilization of trialkylamines in the Ortolev-King reaction.,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 479–483 (1963).

  39. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. VII. 2-Furylglyoxal, 5-nitro-2-furylglyoxal, and their derivatives,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 858–862 (1963).

  40. B. V. Kurgan, S. A. Giller, and A. A. Gruze, “β-Hydroxyethylhydrazides of furancarboxylic acids,” Zh. Obshch. Khim., 2664–2667 (1964).

  41. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. VIII. 2-Furylglyoxylic acid derivatives,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 701–706 (1964).

  42. N. O. Saldabol, A. Ya. Medne, and S. A. Giller, “Synthesis and transformations of furan derivatives. II. Derivatives of 2-amino- and 2-hydrazino-4-(5′-nitro-2′-furyl) thiazoles,” Zh. Obshch. Khim., 34, 1598–1601 (1964).

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  43. G. P. Sokolov, M. G. Voronkov, and S. A. Giller, “Reaction of 2,5-dimethoxytetrahydrofuran with glycols. Synthesis of cyclic diacetals of succinic dialdehyde,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 667–672 (1964).

  44. G. P. Sokolov, S. A. Giller, M. G. Voronkov, “Reaction of organomagnesium compounds with 2,5-dimethoxy-2,5-dihydrofurans,” Dokl. Akad. Nauk SSR, 158, 675–678 (1964).

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  45. K. Venters and S. Hillers, “Functional derivatives of 5-nitro-2-furylpolyalkenes,” in: Nitro Compounds. Proceedings of the International Symposium Held at the Polish Academy of Sciences. Warsaw, Sept. 18–20, 1963, Warsaw-London (1964), pp. 71–79 (Tetrahedron, 20, 1).

  46. S. A. Giller and Ya. A. Kastron, “Method for the preparation of polymers,” USSR Author's Certificate No. 167922; Byul. Izobr., No. 3, 38 (1964).

  47. S. A. Giller and R. Yu. Kalnberg, “Method for the preparation of 3-(5-nitro-2-furfuryli-deneamino)-2-oxazolidone (furazolidone),” USSR Author's Certificate No. 160508; Byul. Izobr., No. 4, 15 (1964).

  48. G. P. Sokolov, M. G. Voronkov, and S. A. Giller, “Method for the preparation of cyclic acetals of succinic and maleic dialdehydes,” USSR Author's Certificate No. 165468; Byul. Izobr., No. 19, 17 (1964).

  49. K. K. Venter, S. P. Korshunov, L. I. Vereshchagin, R. L. Bol 'shedvorskaya, D. O. Lolya, and S. A. Giller, “Synthesis of 5-nitro-2-furyl- and 2-furylpropiolic acids,” Khim. Geterotsikl. Soedin., 616–619 (1965).

  50. S. A. Giller, A. A. Anderson, A. É. Berzinya, and M. V. Shimanskaya, “Research on the alkylation of furan with olefins. VI. Investigation of the products of alkylation of furan with olefins by means of gas-liquid partition chromatography,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 575–578 (1965).

  51. S. A. Giller, L. I. Vereshchagin, K. K. Venter, S. P. Korshunov, V. V. Tsirule, and D. O. Loyla, “2-Furyl and 5-nitro-2-furyl acetylenic ketones,” Dokl. Akad. Nauk SSSR, 164, 99–102 (1965).

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  52. Ya. A. Kastron and S. A. Giller, “Reaction of ethyl β-furylglycidate with ammonia,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 471–477 (1965).

  53. Ya. A. Kastron and S. A. Giller, “Reaction of ethyl β-furylglycidate with aniline and p-toluidine,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 478–481 (1965).

  54. B. V. Kurgan, S. A. Giller, and A. A. Gruze, “N,N-Bis (2-chloroethyl) amides and N,N-bis-(2-chlorethyl)hydrazides of carboxylic acids of the furan series,” Khim. Geterotsikl. Soedin., 11–14 (1965).

  55. G. P. Sokolov and S. A. Giller, “Electrochemical methoxylation of halofurans,” Khim. Geterotsikl. Soedin., 163–170 (1965).

  56. B. V. Kurgan, S. A. Giller, and A. A. Gruze, “Method for the preparation of N,N-bis (2-chlorethyl)hydrazides of furancarboxylic acids,” USSR Author's Certificate No. 169540; Byul. Izobr., No. 7, 27 (1965).

  57. S. A. Giller and A. É. Berzinya, “Research on the alkylation of furan with olefins. VII. Vibrational spectra of alkyl-substituted furans,” Khim. Geterotsikl. Soedin., 487–498 (1968).

  58. B. V. Kurgan and S. A. Giller, “Thioamides of 5-nitrofuran-2-carboxylic and 3-(5′-nitro-2′-furyl) acrylic acids,” Khim. Geterotsikl. Soedin., 323–327 (1966).

  59. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. IX. ω-Ammonium derivatives of methyl 5-nitro-2-furyl ketone,” Khim. Geterotsikl. Soedin., 855–858 (1966).

  60. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. X. 5-Nitro-2-furylglyoxylic acid and its derivatives,” Khim. Geterotsikl. Soedin., 859–862 (1966).

  61. L. I. Vereshchagin, S. P. Korshunov, Ya. A. Éidus, K. K. Venter, and S. A. Giller, “Furylalkynes. VIII. IR spectra and intramolecular interaction in some acetylenic derivatives of furan and thiophene,” Zh. Organ. Khim., 3, 184–189 (1967).

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  62. S. A. Giller, A. Y. Zile, K. K. Venter, S. P. Zaeva, M. A. Al'berta, K. K. Medne, S. K. Germane, and R. Yu. Kalnberg, “Investigations of the fungistatic Properties of derivatives of α, β-unsaturated and polyene aldehydes and ketones of the 5-nitrofuran series,” Izv. Akad. Nauk LatvSSR, No. 12, 99–105 (1967).

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  63. B. V. Kurgan, A. A. Gruze, É. Ya. Lukevits, and S. A. Giller, “2-Haloethyl and 2-haloethylthio esters of carboxylic acids of the furan series,” Khim. Geterotsikl. Soedin., 18–21 (1967).

  64. N. O. Saldabol and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. XI. Monofunctional 5- and 6-(2-furyl)-1,2, 4-triazine derivatives,” Khim. Geterotsikl. Soedin., 14–17 (1967).

  65. N. O. Saldabol, S. A. Giller, L. N. Alekseeva, and B. A. Brizda, “Syntheses in the methyl 2-furyl ketone series. XII. (5-Nitro-2-furyl)-substituted imidazo heterocyclic compounds with a nitrogen atom in common,” Khim.-Farmats. Zh., No. 2, 27–31 (1967).

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  66. N. O. Saldabol, A. Ya. Medke, and S. A. Giller, “Syntheses in the methyl 2-furyl ketone series. XII [XIII]. ω-Derivatives of methyl 5-bromo-2-furyl ketone. XIII [XIV]. ω,ω-Dihalomethyl-2-furyl ketones and their 5-nitro derivatives. 5-Nitro-2-furylglyoxal,” Khim. Geterotsikl. Soedin., 553–556 (1967).

  67. K. K. Venter, S. A. Giller, and V. V. Tsirule, “Method for the preparation of β-(5-nitro-2-furyl)acrolein,” USSR Author's Certificate No. 224530; Byul. Izobr., No. 26, 34 (1968).

  68. L. I. Vereshchagin, R. I. Katkevich, S. A. Giller, K. K. Venter, L. N. Alekseeva, L. V. Kruzmetra, Z. Ya. Zile, and N. P. Glazunova, “Synthesis and antibiotic properties of some nitrofurylacetylenic compounds, ” Khim.-Farmats. Zh., No. 10, 31–34 (1968).

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  69. M. A. Berklava and S. A. Giller, “Alcohols of the nitrofuran series. II. Reduction of α-ethyl-β-(5-nitro-2-furyl) acrolein and 5-(5-nitro-2-furyl)-2,4-pentadienal with sodium borohydride,” Khim. Geterotsikl. Soedin., 12–16 (1967).

  70. A. Ya. Perkone, N. O. Saldabol, and S. A. Giller, “Bromination of 2-amino- and 2-acetamido-4-(2-furyl) thiazoles,” Khim. Geterotsikl. Soedin., 498–500 (1969).

  71. K. K. Venter, S. A. Giller, M. A. Apsite, V. É. Égert, and Z. Ya. Zelmene, “Method for the preparation of 5-nitrofurfurylideneacetylhydrazone or its vinylogs,” USSR Author's Certificate No. 250156; Byul. Izobr., No. 26, (1969).

  72. V. V. Kotetskii, Ya. A. Kharit, L. A. Vol'f, A. I. Meos, S. A. Giller, and K. K. Venter, “Method for the preparation of chemical fibers with disinfectant properties,” USSR Author's Certificate No. 256934; Byul. Izobr., No. 35, 55 (1969).

  73. S. A. Giller, M. V. Shimanskaya, V. É. Égert, and K. K. Venter, “Method for the preparation of water-soluble salts of 1-(5-nitrofurfurylideneamino) hydantoin and its vinylogs,” USSR Author's Certificate No. 274113; Byul. Izobr., No. 21, 28 (1970).

  74. A. A. Lazdyn'sh, K. K. Venter, and S. A. Giller, “Method for the preparation of β-(5-nitro-2-furyl) acrolein,” USSR Author's certificate No. 269926; Byul. Izobr., No. 16, 21 (1970).

  75. N. O. Saldabol and S. A. Giller, “Nitration of 2-acetylfuran and acetophenone oximes,” in: The Chemistry of Heterocyclic Compounds. Collection 2. Oxygen-Containing Heterocycles [in Russian], Riga (1970), pp. 118–121.

  76. N. O. Saldabol and S. A. Giller, “Synthesis and transformations of 5-nitro-2-propionylfuran,” in: The Chemistry of Heterocyclic Compounds. Collection 2. Oxygen-Containing Heterocycles [in Russian], Riga (1970), pp. 122–124.

  77. S. A. Giller, K. K. Venter, M. A. Apsite, V. E. Égert, R. Yu. Kalnberg, and L. V. Kruzmetra, “Method for the preparation of 3-(5′-nitrofurfurylideneamine)hydantoic acid derivatives,” USSR Author's Certificate No. 313435; Byul. Izobr., No. 12, 242 (1972).

  78. N. O. Saldabol, L. L. Zeligman, S. A. Giller, Yu. Yu. Popelis, A. É. Abele, and L. N. Alekseeva, “Nitrosation and bromination of 6-(2′-furyl) imidazo[2,1-b] thiazole and its derivatives,” Khim. Geterotsikl. Soedin., 1353–1358 (1972).

  79. S. A. Giller, L. A. Vol'f, and A. I. Meos, “Method for the modification of fibers and films,” Italian Patent No. 712346 (1966).

  80. S. A. Giller, K. K. Venter, and V. V. Tsirule, “Method for the preparation of β-(5-nitro-2-furyl) acrolein,” Italian Patent No. 733091 (1966); British Patent No. 1109417 (1968).

  81. S. A. Giller, L. A. Vol'f, and A. I. Meos, “Method for the modification of polyvinyl alcohol,” Japanese Patent No. 530039 (1968).

  82. S. A. Giller, M. V. Shimanskaya, V. É. Égert, and K. K. Venter, “Water-soluble alkali metal salts of 1-(5′-nitrofurfurylideneamino) hydantoin and its vinylogs,” British Patent No. 1129195 (1968); French Patent No. 1529664 (1968).

  83. S. A. Giller, L. A. Vol'f, and A. I. Meos, “Treatment of fibers and films,” British Patent No. 1085554 (1968).

  84. S. A. Giller, K. K. Venter, and A. A. Lazdyn'sh, “Treatment of fibers and films,” French Patent No. 1555141 (1968).

  85. S. A. Giller, K. K. Venter, and A. A. Lazdyn'sh, “Improved method for the preparation of β-(5-nitro-2-furyl) acrolein,” British Patent No. 1164588 (1969).

  86. S. A. Giller, M. V. Shimanskaya, V. É. Égert, and K. K. Venter, “Improved method for the preparation of β-(5-nitro-2-furyl) acrolein,” US Patent No. 3531477 (1970).

  87. S. A. Giller, M. V. Shimanskaya, V. É. Égert, and K. K. Venter, “Method for the preparation of water-soluble potassium and sodium salts of hydantoin derivatives,” Swiss Patent No. 498143 (1970).

  88. S. A. Giller, K. K. Venter, and V. V. Tsirule, “Method for the preparation of water-soluble potassium and sodium salts of hydantoin derivatives,” US Patent No. 3491123 (1970).

  89. S. A. Giller, K. K. Venter, and A. A. Lazdyn'sh, “Method for the preparation of water-soluble potassium and sodium salts of hydantoin derivatives,” Swiss Patent No. 507229 (1971); Japanese Patent No. 612033 (1971).

  90. L. A. Vol'f, S. A. Giller, and A. I. Meos, “Method for the modification of fibers and films,” West German Patent No. 1444079 (1973).

  91. N. O. Saldabol, A. Yu. Tsimanis, Yu. Yu. Popelis, and S. A. Giller, “2-(5-Bromo-2-furyl) quinoxaline and 3-(5-bromo-2-furyl)2-quinoxalone,” Khim. Geterotsikl. Soedin., 404–406 (1973).

  92. S. A. Giller, N. O. Saldabol, L. L. Zeligman, “Method for the preparation of 2-(5-nitro-2-furyl) imidazo [1,2-a] pyridine,” USSR Author's Certificate No. 407897; Byul. Izobr., No. 47, 82 (1973).

  93. S. A. Giller, N. O. Saldabol, and A. Yu. Tsimanis, “Method for the preparation of 3-(5-nitro-2-furyl)2-quinoxalone,” USSR Author's Certificate No. 410015; Byul. Izobr., No. 1, 81 (1974).

  94. N. O. Saldabol, A. Yu. Tsimanis, S. A. Giller, Yu. Yu. Popelis, L. N. Alekseeva, A. Ya. Zile, and A. K. Yalynskaya, “Derivatives of 5-nitro-2-furylglyoxal and its analogs,” Khim.-Farmats. Zh., No. 8, 12–16 (1974).

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  95. D. O. Lolya, K. K. Venter, É. É. Liepin'sh, and S. A. Giller, “Nitration of furan derivatives with acetyl nitrate. I. Investigation of the products of nitration of methyl furan-2-carboxylate,” Khim. Geterotsikl. Soedin., 883890 (1975).

II. Chemistry of Ethyleneimine

  1. M. Yu. Lidak and S. A. Giller, “Some reactions of ethyleneimine. I. Reaction of ethyleneimine with aliphatic and carbocyclic aldehydes and ketones,” Izv. Akad. Nauk LatvSSR, No. 5, 99–108 (1961).

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  2. M. Yu. Lidak and S. A. Giller, “Some reactions of ethyleneimine. II. Reaction of ethyleneimine with furfural, benzaldehyde, and their derivatives,” Izv. Akad. Nauk LatvSSR, No. 7, 49–58 (1961).

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  3. M. Yu. Lidak and S. A. Giller, “Some reactions of ethyleneimine. III. Reaction of ethyleneimine with unsaturated aldehydes,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 81–88 (1961).

  4. M. Yu. Lidak and S. A. Giller, “Some reactions of ethyleneimine. IV. Reaction of ethyleneimine with substituted furancarboxylic acid chlorides,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 211–216 (1961).

  5. M. Yu. Lidak and S. A. Giller, “New carcinostatic derivatives of ethyleneimine. Study of the reaction of ethyleneimine with derivatives containing carbonyl and carboxyl functions,” in: Methods for the Synthesis of and Search for Antitumorigenic Preparations [in Russian], Moscow (1962), pp. 193–202.

  6. S. A. Giller, A. V. Eremeev, M. Yu. Lidak, and V. A. Pestunovich, “Chemistry of ethyleneimine. I. N-Aminoethyleneimine. II. Mechanism of the oxidative transformation of N-aminoethyleneimine,” Khim. Geterotsikl. Soedin., 815–822 (1968).

  7. S. A. Giller, A. V. Eremeev, and M. Yu. Lidak, “Chemistry of ethyleneimine. III. Reaction of N-aminoethyleneimine with the simplest aliphatic aldehydes and acrolein,” Khim. Geterotsikl. Soedin., 3–7 (1970).

  8. S. A. Giller, A. V. Eremeev, M. Yu. Lidak, and V. A. Pestunovich, “Chemistry of ethyleneimine. IV. Heterolysis of the ring of N-aminoethyleneimine under the influence of sulfonyl halides,” Khim. Geterotsikl. Soedin., 8–11 (1970).

  9. S. A. Giller, A. V. Eremeev, M. Yu. Lidak, and V. A. Kholodnikov, “Chemistry of ethyleneimine. V. Derivatives of the sulfate ester of β-hydroxyethylhydrazine and their conversion under the conditions of the Wenker synthesis. VI. N,N-Ethylenehydrazones of ketones,” Khim. Geterotsikl. Soedin., 466–474 (1970).

  10. S. A. Giller, A. V. Eremeev, and M. Yu. Lidak. V. A. Pestunovich, É. É. Liepin'sh, and I. Ya. Kalvin'sh, “Chemistry of ethyleneimine. VII. Pyramidal stability of N-aminoethyleneimine derivatives,” Khim. Geterotsikl. Soedin., 45–48 (1971).

  11. S. A. Giller, A. V. Eremeev, M. Yu. Lidak, V. A. Kholodnikov, and V. A. Pestunovich, “Chemistry of ethyleneimine. VIII. Synthesis and properties of 2-alkyl-substituted 1,3-diazabicyclo [3.1.0] hexane,” Khim. Geterotsikl. Soedin., 607–609 (1971).

  12. S. A. Giller, A. V. Eremeev, V. A. Pestunovich, M. Yu. Lidak, R. G. Kostyanovskii, O. A. Pan'shin, Z. E. Samoilova, and I. I. Chervin, “Phenomenon of the configurational stability of trivalent nitrogen in nonbridged structures,” Byul. Izobr., No. 24, 3 (1972).

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  13. S. A. Giller, M. Yu. Lidak, A. V. Eremeev, and V. A. Kholodnikov, “Chemistry of ethyleneimine. IX. Preparation and properties of 2-aryl-substituted 1,3-diazabicyclo [3.1.0]-hexanes,” Khim. Geterotsikl. Soedin., 483–484 (1972).

  14. S. A. Giller, É. É. Liepin'sh, V. A. Pestunovich, A. V. Eremeev, and V. A. Kholodnikov, “1H and 13C NMR spectra of N-aminoethyleneimine hydrazones,” Khim. Geterotsikl. Soedin., 571–573 (1975).

  15. S. A. Giller, R. S. Él'kinson, and A. V. Eremeev, “Conjugation of the aziridine and benzene rings in a number of p-substituted N-phenylethyleneimines,” Khim. Geterotsikl. Soedin., 70–72 (1975).

  16. S. A. Giller, A. V. Eremeev, D. A. Tikhomirov, and É. É. Liepin'sh, “Synthesis of arylhydrazones of 1-amino-2-arylethyleneimines,” Khim. Geterotsikl. Soedin., 426–429 (1975).

  17. S. A. Giller, É. É. Liepin'sh, V. A. Pestunovich, A. V. Eremeev, and V. A. Kholodnikov, “Chemistry of ethyleneimine. X. PMR spectra of substituted 1,3-diazabicyclo [3.1.0] hexanes,” Khim. Geterotsikl. Soedin., 928–936 (1975).

  18. S. A. Giller, A. V. Eremeev, V. A. Kholodnikov, and É. É. Liepin'sh, “Chemistry of ethyleneimine. XI. Addition of 2-aminomethylethyleneimine to an activated carbon-carbon double bond,” Khim. Geterotsikl. Soedin., 1212–1216 (1975).

  19. S. A. Giller, É. É. Liepin'sh, A. V. Eremeev, I. Ya. Kalvin'sh, V. A. Kholodnikov, and V. A. Pestunovich, “Configuration of 2-substituted 1-aminoethyleneimines,” 1337–1339 (1975).

  20. S. A. Giller, A. V. Eremeev, I. Ya. Kalvin'sh, and É. É. Liepin'sh, “Chemistry of ethyleneimine. XII. Transformations of 1-chloro-2-cyano-(2,2-dimethylhydrazino) ethane in the presence of sodium hydride,” Khim. Geterotsikl. Soedin., 1503–1505 (1975).

  21. S. A. Giller, A. V. Eremeev, I. Ya. Kalvin'sh, É. É. Liepin'sh, and V. G. Semenikhina,” Derivatives of 1-H-aziridine-2-carboxylic acid,” Khim. Geterotsikl. Soedin., 1625–1631 (1975).

  22. S. A. Giller, Ya. Ya. Bleidelis, A. A. Kemme, A. V. Eremeev, and V. A. Kholodnikov, “Crystalline and molecular structure of 2-(o-bromophenyl) -1,3-diazabicyclo [3.1.0] hexane,” Zh. Strukt. Khim., 3, 411–415 (1975).

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  23. S. Giller (Hiller), Ya. Bleidelis, A. Kemme, and A. Eremeev (Eremeyev), “X-ray crystal and molecular structure determination of a novel bicyclic system — 2-β-bromophenyl-1, 3-diazabicyclo [3. 1.0]hexane,” Chem. Commun., 130 (1975).

III. Chemistry of Five- and Six-Membered Nitrogen-Containing Heterocycles

  1. M. Yu. Lidak, S. A. Giller, and N. N. Naumenko, “Preparation of isonicotinic acid from the light (β-picoline) fraction of pyridine bases,” Izv. Akad. Nauk LatvSSR, No. 12, 83–88 (1953).

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  2. É. É. Dunkel' and S. A. Giller, “Preparation of 1, 2-dihydropyridazine-3,6-dione,” Izv. Akad. Nauk LatvSSR, No. 2, 105–108 (1954).

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  3. Kh. M. Vasserman and S. A. Giller, “Structure and properties of some 3,6-disubstituted pyridazines,” Izv. Akad. Nauk LatvSSR, No. 5, 87–92 (1958).

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  4. Kh. M. Vasserman, S. A. Giller, and A. A. Avot, “Preparative synthesis of new ganglion blockers — pentapyrrolidinium and tetrapiperidinium salts,” Izv. Akad. Nauk LatvSSR, No. 5, 79–86 (1958).

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  5. M. Yu. Lidak, S. A. Giller, and N. N. Naumenko, “Preparation of isonicotinic acid from the light (β-picoline) fraction of pyridine bases,” in: Tubazid [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1958), pp. 9–17.

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  6. G. P. Sokolov, and S. A. Giller, “Method for the preparation of substituted amides and hydrazides of pyridazine-3-carboxylic acid,” USSR Author's Certificate No. 134269; Byul. Izobr., No. 24, 16 (1960).

  7. L. Ya. Avota and S. A. Giller, “Method for the preparation of 1-phenyl-4,5-dichloro-6-pyridazone,” USSR Author's Certificate No. 172335; Byul. Izobr., No. 13, 22 (1965).

  8. S. A. Giller and L. Ya. Avota, “Method for the preparation of 1-phenyl-4-amino-5-chloro-6-pyridazone,” USSR Author's Certificate No. 172813; Byull. Izobr., No. 14, 29 (1965).

  9. S. A. Giller, K. K. Venter, G. D. Tirzit, Kh. I. Girshovich, Z. G. Fridman, and S. G. Fridlender, “Method for the preparation of the cyclic hydrazide of maleic acid,” USSR Author's Certificate No. 174631; Byul. Izobr., No. 18, 27 (1965).

  10. L. Ya. Avota, N. Ya. Ozolinya, and S. A. Giller, “Research in the 1-phenyl-6-pyridazone series. I. Reaction of 1-phenyl-4,5-dichloro-6-pyridazone with ammonium hydroxide,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 347–352 (1967).

  11. S. A. Giller and L. Ya. Avota, “Dipyridazo[4,5-b∶4,5-e]-1,4-dithiynes and dipyridazo sulfides,” Khim. Geterotsikl. Soedin., 572 (1967).

  12. G. P. Sokolov and S. A. Giller, “Synthesis of some bis heterocycles of the pyridazine series,” Khim. Geterotsikl. Soedin., 556–559 (1967).

  13. S. A. Giller, L. Ya. Avota, and N. Ya. Ozolinya, “Preparation of 1-phenyl-4,5-dichloro-6-pyridazone,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 348–352 (1968).

  14. R. A. Zhuk, Ya. A. Éidus, and S. A. Giller, “Synthesis, structure, and spectra of 6-(2-furylpolyene) derivatives of 5-nitrouracil,” Khim. Geterotsikl. Soedin., 1111–1115 (1968).

  15. N. O. Saldabol, G. Ya. Zarinya, and S. A. Giller, “6-(2-Furyl)imidazo [2,1-b]thiazole and its derivatives,” Khim. Geterotsikl. Soedin., 178–180 (1968).

  16. S. A. Giller, G. Ya. Dubur, Ya. R. Uldrikis, G. D. Tirzit, A. R. Val'dman, I. M. Zakharchenko, Ya. Ya. Spruzh, V. E. Ronis, and A. A. Makarov, “Method for the preparation of 3,5-dicarbonyl derivatives of 2,6-dimethyl-1,4-dihydropyridines,” USSR Author's Certificate No. 300465; Byul. Izobr., No. 13, 95 (1971).

  17. N. O. Saldabol, L. L. Zeligman, and S. A. Giller, “Aminomethylation of 2-(2-furyl)-imidazo[1,2-a/pyridine,” Khim. Geterotsikl. Soedin., 818–821 (1971).

  18. N. O. Saldabol, L. L. Zeligman, and S. A. Giller, “Application of the King method for the synthesis of imidazo[1,2-a/pyridines,” Khim. Geterotsikl. Soedin., 860–861 (1971).

  19. S. A. Giller, A. A. Lazdyn'sh, D. Ya. Snikere, A. K. Veinberg, I. L. Knunyants, L. S. German, and N. B. Kozmina, “Method for the preparation of 5-fluorouracil,” USSR Author's Certificate No. 322053; Byul. Izobr., No. 32, 186 (1972).

  20. N. O. Saldabol, S. A. Giller, L. N. Alekseeva, and I. V. Dipan, “3-Nitro derivatives of 2-(2-furyl) indolizine and 2-(furyl)imidazo[1,2-a/pyridine and its substituted derivatives,” Khim.-Farmats. Zh., No. 6, 16–19 (1972).

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  21. S. A. Giller and L. Ya. Avota, “Method for the preparation of N1-tetrahydropyranyl- and N1-tetrahydrofuranyl-3-hydroxy-6-pyridazones,” USSR Author's Certificate No. 382629; Byul. Izobr., No. 23, 61 (1973).

  22. L. Ya. Avota, I. V. Turovskii, and S. A. Giller, N1-Tetrahydrofuranyl- and N1-tetrahydropyanyl-3-hydroxy-6-pyridazones,” Khim. Geterotsikl. Soedin., 1545–1547 (1973).

  23. N. O. Saldabol, L. L. Zeligman, and S. A. Giller, “β-Substituted 2-vinylimidazo[1,2-a/-pyridines from saturated ketones,” Khim. Geterotsikl. Soedin., 137–141 (1973).

  24. A. D. Voitenko, Ya. A. Kastron, É. É. Liepin'sh, and S. A. Giller, “Alkylation of 3-isoxazolidone,” Khim. Geterotsikl. Soedin., 3–7 (1973).

  25. A. D. Voitenko, Ya. A. Kastron, and S. A. Giller, “Mechanism of the alkylation of isoxazolidone,” Khim. Geterotsikl. Soedin., 898–901 (1973).

  26. N. O. Saldabol, A. Yu. Tsimanis, and S. A. Giller, “N-Oxides in the synthesis of arylglyoxylic acids,” Zh. Organ. Khim., 5, 1059–1063 (1974).

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  27. S. A. Giller, L. Ya. Avota, and A. A. Lazdyn'sh, “Method for the preparation of 1-phenyl-4,5-dichloro-6-pyridazone,” USSR Author's Certificate No. 436055; Byul. Izobr., No. 26, 67 (1974).

  28. S. A. Giller, A. V. Eremeev, I. Ya. Kalvin'sh, É. É. Liepin'sh, and D. A. Tikhomirov, “Reaction of α-chloroacrylonitrile with hydrazines,” Khim. Geterotsikl. Soedin., 246–249 (1975).

  29. S. A. Giller, G. Ya. Dubur, Ya. R. Uldrikis, A. R. Val'dmans, I. M. Zakharchenko, Ya. Ya. Spruzh, V. E. Ronis, A. A. Makarova, and G. D. Tirzit, “Method for the preparation of 3,5-dicarbonyl derivatives of 2,6-dimethyl-1,4-dihydropyridines,” French Patent No. 7026988 (1972); British Patent No. 1294650 (1972); US Patent No. 3883673 (1975).

  30. L. Ya. Avota, V. A. Pestunovich, and S. A. Giller, “Silylation of 6-pyridazone derivatives,” Khim. Geterotsikl. Soedin., 990–996 (1976).

IV. Analogs of Nucleosides and Nucleotides

  1. S. A. Giller, “State and tasks of scientific research on the synthesis of physiologically active polymeric substances,” Paper presented at the All-Union Conference on Physiologically Active Polymeric Substances [in Russian], Riga (1962), pp. 1–10.

  2. S. A. Giller, R. A. Zhuk, and M. Yu. Lidak, “Analogs of pyrimidine nucleosides. I. N1-(α-Furanidyl) derivatives of natural pyrimidine bases and their antimetabolites,” Dokl. Akad. Nauk SSSR, 176, 332–335 (1967).

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  3. S. A. Giller, R. A. Zhuk, and Ya. G. Nashatyr', Analogs of pyrimidine nucleosides. II. N1-(α-Butyrolactono) derivatives of 5-substituted uracils,” Khim. Geterotsikl. Soedin., 557–558 (1968).

  4. D. Ya. Sniker, R. A. Zhuk, É. I. Stankevich, G. Ya. Dubur, and S. A. Giller, “Analogs of pyrimidine nucleosides. III. N1-(α-Furanidyl)-5,6-dihydrouracil derivatives,” Khim. Geterotsikl. Soedin., 170–172 (1969).

  5. S. A. Giller, M. Yu. Lidak, R. A. Zhuk, A. É. Berzinya, K. Ya. Pets, I. N. Getsova and É. I. Bruk, “Analogs of pyrimidine nucleosides. IV. Silyl method for the preparation of N1-(α-furanidyl)- and N1-(α-pyranidyl) derivatives of uracils and 6-azauracils,” Khim. Geterotsikl. Soedin., 375–377 (1969).

  6. S. A. Giller, R. A. Zhuk, and M. Yu. Lidak, “Method for the preparation of N-substituted furanidylpyrimidines,” USSR Author's Certificate No. 272307; Byul. Izobr., No. 19, 28 (1970).

  7. S. A. Giller, R. A. Zhuk, M. Yu. Lidak, A. É. Berzinya, I. N. Getsova, K. Ya. Pets, and É. I. Bruk, “Method for the preparation of N1-furanidyl- or N1-pyranidyl derivatives of 5-substituted uracils or 6-azauracils,” USSR Author's Certificate No. 287952; Byul. Izobr., No. 36, 32 (1970).

  8. R. A. Zhuk, Yu. Yu. Popelis, and S. A. Giller, “Analogs of pyrimidine nucleosides. V. UV spectra and protolysis constants of N1-(2′-furanidyl)- and N1-(α-butyrolactono)-5-substituted uracils,” Khim. Geterotsikl. Soedin., 546–549 (1970).

  9. R. A. Zhuk, A. É. Berzinya, G. G. Volynkina, and S. A. Giller, “Analogs of pyrimidine nucleosides. VI. Kinetics of the acid hydrolysis of N1-(2′-furanidyl)- and N1-(2′-pyranidyl) derivatives of uracil, thymine, and 5-fluorouracil,” Khim. Geterotsikl. Soedin., 550–553 (1970).

  10. S. A. Giller, A. Ya. Perkone, I. N. Getsova, A. B. Rozenblit, and V. E. Golender, “N1-(2-Furoylmethyl)- and N1-(5-nitro-2-furoylmethyl) derivatives of uracil and 5-substituted uracils,” Khim. Geterotsikl. Soedin., 1268–1270 (1971).

  11. S. A. Giller, R. A. Zhuk, A. É. Berzinya, and L. A. Sherinya, “Method for the preparation of N1-(butyrolactono-γ-methylene)-5-substituted uracils,” USSR Author's Certificate No. 348563; Byul. Izobr., No. 25, 91 (1972).

  12. S. A. Giller, R. A. Zhuk, M. Yu. Lidak, and A. A. Ziderman, “N1-(2′-Furanidyl) derivatives of 5-substituted uracils,” US Patent No. 3635946 (1972).

  13. S. A. Giller, I. N. Goncharova, I. N. Getsova, L. I. Mironova, É. I. Bruk, G. F. Nazarova, and L. N. Petrulyanis, “Analogs of purine nucleosides and purine mono- and polynucleotides. I. Synthesis of phosphate esters of 6-substituted 9-(α,ω-dihydroxy-2-alkyl)purines,” Khim. Geterotsikl. Soedin., 1674–1679 (1974).

  14. S. A. Giller, I. N. Getsova, I. N. Goncharova, L. N. Petrulyanis, L. I. Mironova, G. F. Nazarova, and É. I. Bruk, “Analogs of purine nucleosides and purine mono- and polynucleotides. II. Substituted α-(9-purinyl)-γ-butyrolactones,” Khim. Geterotsikl. Soedin., 1680–1683 (1974).

  15. S. A. Giller, I. N. Goncharova, I. N. Getsova, Yu. A. Benders, and Ya. P. Stradyn', “Analogs of purine nucleosides and purine mono- and polynucleotides. III. Intermolecular and intramolecular interactions in 6-substituted 9-(α,ω-dihydroxyalkyl)purines,” Khim. Geterotsikl. Soedin., 1684–1689 (1974).

  16. S. A. Giller, R. A. Zhuk, A. É. Berzinya, L. T. Kaulinya, and L. Ya. Sherin', “Analogs of pyrimidine nucleosides. VII. 5-Substituted N1-(1,4-dihydroxy-2-butyl)- and N1-(2,5-dihydroxy-1-pentyl)uracils,” Khim. Geterotsikl. Soedin., 1662–1665 (1974).

  17. R. A. Zhuk, L. A. Sherin', É. É. Liepin'sh, and S. A. Giller, “Analogs of pyrimidine nucleosides. VIII. Synthesis and properties of substituted α-(1-uracilyl)-γ-methyl-γ-butyrolactones and N1-(1,4-dihydroxy-2-pentyl)uracils,” Khim. Geterotsikl. Soedin., 1666–1670 (1974).

  18. S. A. Giller, L. A. Sherin', R. A. Zhuk, and A. É. Berzinya, “Analogs of pyrimidine mono- and polynucleotides. I. Diphosphates of N1-(1,4-dihydroxy-2-butyl) derivatives of uracil and thymine,” Khim. Geterotskikl. Soedin., 1671–1673 (1974).

  19. S. A. Giller and Z. A. Shomshtein, “Synthesis of N1-(3-furanidyl)thymine,” Khim. Geterotsikl. Soedin., 1700–1701 (1974).

  20. S. A. Giller, I. N. Goncharova, I. N. Getsova, L. N. Petrulyanis, L. I. Mironova, E. I. Bruk, and É. É. Liepin'sh, “Analogs of purine nucleosides and purine mono- and polynucleotides. IV. Acylation of 6-substituted 9-(α,ω)-dihydroxy-2-alkyl)purines,” Khim. Geterotsikl. Soedin., 132–137 (1975).

  21. S. A. Giller, T. A. Popova, and Z. A. Shomshtein, “Analogs of pyrimidine mono- and polynucleotides. II. Phosphorylation of N1-(1,4-dihydroxy-2-butyl)thymine,” Khim. Geterotsikl. Soedin., 401–408 (1975).

  22. S. A. Giller, Z. A. Shomshtein, and T. A. Popova, “Analogs of pyrimidine mono- and polynucleotides. III. Analogs of oligothymidylic acid,” Khim. Geterotsikl. Soedin., 409–416 (1975).

  23. S. A. Giller, Z. A. Shomshtein, and T. A. Popova, “Analogs of pyrimidine mono- and polynucleotides. IV. Reaction of a polythymidylic acid analog based on N1-(1,4-dihydroxy-2-butyl)-thymine with polyadenylic acid,” Khim. Geterotsikl. Soedin., 416–421 (1975).

  24. S. A. Giller, Z. A. Shomshtein, and T. A. Popova, “Analogs of pyrimidine mono- and polynucleotides. V. Synthesis of models of di- and trinucleotides by thermal polycondensation,” Khim. Geterotsikl. Soedin., 540–543 (1975).

  25. S. A. Giller, R. A. Zhuk, A. É. Berzinya, and L. T. Kaulinya, “Analogs of pyrimidine nucleosides. IX. N1-Dihydroxyalkyl derivatives of cytosine,” Khim. Geterotsikl. Soedin., 694–699 (1975).

  26. S. A. Giller, É. Ya. Gren, Z. A. Shomshtein, R. A. Zhuk, V. M. Berzin', N. P. Pumpen, and G. F. Rozental', “Synthesis and properties of analogs of polynucleotides based on N1-(1,4-dihydroxy-2-butyl)thymine,” Dokl. Akad. Nauk SSSR, 221, 473–476 (1975).

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  27. S. A. Giller, R. A. Zhuk, A. É. Berzin', L. A. Sherin', and A. A. Zidermane, “Method for the preparation of N1-(α-butyrolactono)- and N1-(α-valerolactono)-5-substituted uracils,” British Patent No. 1386205 (1975).

  28. S. A. Giller, R. A. Zhuk, A. É. Berzin', and L. A. Sherin', “Method for the preparation of N1-(dihydroxyalkyl) derivatives of 5-substituted uracils,” BritishPatent No. 1393863 (1975).

  29. Z. A. Shomshtein and S. A. Giller, “Model analogs of nucleic acids,” Khim. Geterotsikl. Soedin., 27–42 (1976).

V. Modified Antibiotics

  1. G. I. Kleiner, S. A. Giller, G. P. Sokolov, and A. D. Kosyanich, “Method for the preparation of benzylpenicillin diethylaminoethyl ester hydriodide,” USSR Author's Certificate No. 122847; Byul. Izobr., No. 19, 33 (1959).

  2. Ya. A. Kastron, G. A. Veinberg, R. A. Gavar, and S. A. Giller, “2,4-Dimethyl-5-nitrofuran-3-carboxylic acid and its derivatives,” Khim. Geterotsikl. Soedin., 863–867 (1966).

  3. Ya. A. Kastron, G. A. Veinberg, and S. A. Giller, “Semisynthetic nitrofuran penicillins,” Dokl. Akad. Nauk SSSR, 175, 88–91 (1967).

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  4. G. A. Veinberg, Ya. A. Kastron, and S. A. Giller, “Semisynthetic penicillins of the furfurylidene- and 5-nitrofurfurylidenehomophthalic series,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 55–63 (1968).

  5. Ya. A. Kastron, G. A. Veinberg, L. V. Kruzmetra, A. Ya. Zile, and S. A. Giller, “Semisynthetic nitrofuran penicillins and their antimicrobial properties,” in: Semisynthetic Penicillins [in Russian], Moscow (1969), pp. 40–43.

  6. G. A. Veinberg, Ya. A. Kastron, and S. A. Giller, “Hydrolysis of furan and 5-nitrofuran penicillins by the penicillinase Bacillus licheniformis,” Khim. Geterotsikl. Soedin., 295–298 (1971).

  7. A. D. Voitenko, Ya. A. Kastron, K. K. Medne, and S. A. Giller, “Reaction of 2,5-diformylfuran with D-cycloserine,” Khim.-Farmats. Zh., 24–26 (1972).

  8. Ya. A. Kastron, V. V. Novikova, É. É. Liepin', and S. A. Giller, “Synthesis of derivatives of oleandomycin aminohydrin,” Khim. Geterotsikl. Soedin., 168–171 (1974).

  9. É. A. Rudzit, G. Kh. Khisamutdinov, D. A. Kulikova, T. P. Radkevich, L. I. Lisitsa, Ya. A. Kastron, G. A. Veinberg, and S. A. Giller, “Some correlations between structure and effect in a number of furan derivatives of 6-aminopenicillanic acid,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 104–109 (1974).

VI. Catalytic Synthesis of Heterocyclic Compounds

  1. S. A. Giller and M. V. Tarvid, “Catalytic vapor-phase oxidation of furan by air oxygen,” Izv. Akad. Nauk LatvSSR, No. 11, 89–92 (1952).

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  2. M. V. Tarvid, S. A. Giller, and P. F. Kalnin'sh, “Catalytic oxidation of furfural in the vapor-gas phase by air oxygen,” Izv. Akad. Nauk LatvSSR, No. 11, 57–88 (1952).

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  3. A. Ya. Karmil'chik and S. A. Giller, “Isolation of furan from the contact gases formed in the vapor-phase decarbonylation of furfural by means of organic solvents,” Izv. Akad. Nauk LatvSSR, No. 8, 105–108 (1956).

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  4. A. Ya. Karmil'chik and S. A. Giller, “Modification of an oxide catalyst for the vaporphase decarbonylation of furfural by means of alkali-metal salts,” in: Problems in the Chemistry of Timber and Wood [in Russian], Riga (1957), pp. 272–281.

  5. A. Ya. Karmil'chik and S. A. Giller, “Vapor-phase decarbonylation of furfural over a catalyst obtained from a mixture of aluminum, chromium, zinc, and maganese oxides,” in: Problems in the Chemistry of Timber and Wood [in Russian], Riga (1957), pp. 251–269.

  6. S. A. Giller and A. Ya. Karmil'chik, “Method for the isolation of furan from the contact gases formed in the vapor-phase decarbonylation of furfural,” USSR Author's Certificate No. 110962; Byul. Izobr., No. 1, 25 (1958).

  7. S. A. Giller, “Decarbonylation of furfural over quicklime,” in: Problems in the Utilization of Pentosan-Containing Raw Material [in Russian], Riga (1958), pp. 299–308.

  8. S. A. Giller, A. Ya. Karmil'chik, V. I. Lutkova, and L. D. Pertsov, “Method for the preparation of a catalyst for the vapor-phase preparation of furan from furfural,” USSR Author's Certificate No. 115346; Byul. Izobr., No. 10, 26 (1958).

  9. A. Ya. Karmil'chik and S. A. Giller, “Study of the vapor-phase decarbonylation of furfural over a catalyst obtained from a mixture of aluminum, chromium, zinc, and maganese oxides,” in: Problems in the Utilization of Pentosan-Containing Raw Material [in Russian], Riga (1958), pp. 327–339.

  10. M. V. Shimanskaya and S. A. Giller, “Effect of the composition of vanadium catalysts on their activity in the vapor-phase oxidation of furfural,” Izv. Akad. Nauk LatvSSR, No. 9, 93–102 (1960).

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  11. V. A. Slavinskaya, M. V. Shimanskaya, S. A. Giller, and I. I. Ioffe, “Kinetics of the vapor-phase catalytic oxidation of furfural,” Kinet. Katal., No. 2, 252–257 (1961).

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  12. A. Ya. Karmil'chik and S. A. Giller, “Mechanism of the vapor-phase decarbonylation of furfural over oxide catalysts,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 559–562 (1962).

  13. L. Ya. Leitis, M. V. Shimanskaya, and S. A. Giller, “Effect of dimerization of formaldehyde in the vapor-gas phase over vanadium catalyts,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 455–461 (1962).

  14. S. A. Giller, I. I. Ioffe, V. A. Slavinskaya, and M. V. Shimanskaya, “Method for the preparation of maleic anhydride,” USSR Author's Certificate No. 151684; Byul. Izobr., No. 22, 26 (1962).

  15. S. A. Giller, A. A. Avot, I. I. Ioffe, V. A. Slavinskaya, and M. V. Shimanskaya, “Method for the preparation of maleic anhydride,” USSR Author's Certificate No. 158572; Byul. Izobr., No. 22, 11 (1963).

  16. A. A. Anderson, S. A. Giller, M. Ya. Zavitskaya, I. I. Ioffe, D. K. Kurgan, and M. V. Shimanskaya, “Method for the preparation of piperazine,” USSR Author's Certificate No. 166033; Byul. Izobr., No. 21, 15 (1964).

  17. A. Ya. Karmil'chik and S. A. Giller, “Semiconductor catalysts for the decarbonylation of furfural,” in: Scientific Foundations of the Selection and Production of Catalysts [in Russian], Novosibirsk (1964), pp. 255–261.

  18. A. A. Avot, S. A. Giller, G. V. Glemite, M. K. Sile, and M. V. Shimanskaya, “Method for the preparation of maleic anhydride,” USSR Author's Certificate No. 175500; Byul. Izobr., No. 20, 21 (1965).

  19. A. A. Anderson, D. K. Kurgan, S. A. Giller, and M. V. Shimanskaya, “Dehydration of ethanolamine on oxide catalysts,” in: Piperazine [in Russian], Riga (1965), pp. 25–39.

  20. S. A. Giller, M. V. Shimanskaya, B. É. Gofman, and A. A. Anderson, “Deamination of diethylenetriamine at atmospheric pressure,” in: Piperazine [in Russian], Riga (1965), pp. 41–54.

  21. S. A. Giller, A. Ya. Karmil'chik, and M. V. Shimanskaya, “Method for the preparation of α-methylfuran,” USSR Author's Certificate No. 186500; Byul. Izobr., No. 19, 36 (1966).

  22. A. A. Anderson, S. P. Yurel', M. V. Shimanskaya, and S. A. Giller, “Vapor-phase catalytic determination of polyfunctional amines,” Dokl. Akad. Nauk SSSR, 169, 1332–1334 (1966).

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  23. A. Ya. Karmil'chik, G. É. Domburg, M. V. Shimanskaya, and S. A. Giller, “Thermographic study of one of the steps in the production of catalysts used for the preparation of furan and α-methylfuran,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 751–753 (1967).

  24. A. Ya. Karmil'chik, V. V. Stonkus, S. A. Giller, and M. V. Shimanskaya, “Vapor-phase decarbonylation of 5-methylfurfural over mixed-oxide catalysts,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 585–590 (1967).

  25. A. Ya. Karmil'chik and S. A. Giller, “Method for the preparation of a catalyst for the vapor-phase preparation of furan,” USSR Author's Certificate No. 191490; Byul. Izobr., No. 4, 21 (1967).

  26. A. A. Avot, S. A. Giller, D. P. Kikust, D. R. Kreile, É. É. Paulane, V. A. Slavinskaya, M. V. Shimanskaya, and D. Ya. Églite, “Method for the preparation of maleic anhydride,” USSR Author's Certificate No. 234384; Byul. Izobr., No. 18, 194 (1969).

  27. S. A. Giller, M. V. Shimanskaya, B. É. Gofman, and A. A. Lazdyn'sh, “Method for the liquid-phase catalytic deaminocyclization of diethylenetriamine or a mixture of diethylenetriamine with triethyletetramine and tetraethylenepentamine,” USSR Author's Certificate No. 271525; Byul. Izobr., No. 18, 26 (1970).

  28. A. Ya. Karmil'chik and S. A. Giller, “Method for the preparation of a catalyst for the synthesis of furan by vapor-phase decarbonylation of furfural,” USSR Author's Certificate No. 305906; Byul. Izobr., No. 19, 23 (1971).

  29. S. A. Giller, M. V. Shimanskaya, B. É. Gofman, and A. A. Lazdyn'sh, “Method for the liquid-phase catalytic diaminocyclization of ethylenediamine, diethylenetriamine, and higher oligomers of ethylenediamine,” USSR Author's Certificate No. 311915; Byul. Izobr., No. 25, 99 (1971).

  30. A. Ya. Karmil'chik and S. A. Giller, “Mechanism of the vapor-phase catalytic decarbonylation of furan aldehydes,” in: Heterogeneous Catalysis in Reactions for the Preparation and Conversion of Heterocyclic Compounds [in Russian], Riga (1971), pp. 35–60.

  31. A. Ya. Karmil'chik, V. V. Stonkus, and S. A. Giller, “Catalytic decarbonylation of mixtures of methylfurfural and furfural,” in: Heterogeneous Catalysis in Reactions for the Preparation and Conversion of Heterocyclic Compounds [in Russian], Riga (1971), pp. 61–67.

  32. M. V. Shimanskaya, S. A. Giller, and I. I. Ioffe, “Vapor-phase catalytic oxidation of furan compounds,” in: Heterogeneous Catalysis in Reactions for the Preparation and Conversion of Heterocyclic Compounds [in Russian], Riga (1971), pp. 5–24.

  33. M. V. Shimanskaya, B. É. Gofman, A. A. Lazdyn'sh, and S. A. Giller, “Catalytic deaminocyclization of polyfunctional amines in the liquid phase,” in: Heterogeneous Catalysis in Reactions for the Preparation and Conversion of Heterocyclic Compounds [in Russian], Riga (1971), pp. 185–194.

  34. A. Ya. Karmil'chik, V. V. Stonkus, and S. A. Giller, “Research on the vapor-phase catalytic conversion of γ-butyrolactone,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 167–173 (1972).

  35. S. A. Giller, V. A. Slavinskaya, I. A. Milman, É. E. Dzilyuma, D. R. Kreile, D. Ya. Églite, M. V. Shimanskaya, and A. K. Strautin', “Method for the vapor-phase catalytic oxidation of furan to maleic anhydride,” USSR Author's Certificate No. 406828; Byul. Izobr., No. 46, 67 (1973).

  36. S. A. Giller, É. E. Dzilyuma, V. A. Slavinskaya, I. A. Milman, I. I. Geiman, D. R. Kreile, and G. P. Sokolov, “Method for the preparation of maleic anhydride,” USSR Author's Certificate No. 385957; Byul. Izobr., No. 26, 82 (1973).

  37. S. A. Giller, and M. V. Shimanskaya, “Mechanism of the catalytic reactions in the oxidation of furan and pyridine compounds,” in: Mechanisms and Kinetics of Heterogeneous Reactions [in Russian], Nauka, Moscow (1973), pp. 47–55.

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  38. S. A. Giller, A. Ya. Karmil'chik, V. V. Stonkus, É. Kh. Korchagova, Zh. G. Baikova, and M. V. Shimanskaya, “Method for the preparation of methyl propyl ketone,” USSR Author's Certificate No. 386906; Byul. Izobr., No. 27, 61 (1973).

  39. A. Ya. Karmil'chik, V. V. Stonkus, M. V. Shimanskaya, and S. A. Giller, “Vapor-phase conversion of ethanol over a promoted chromium-zinc-manganese catalyst,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 421–426 (1974).

  40. S. A. Giller, V. I. Gryaznov, L. F. Pavlova, L. F. Bulenkova, Ya. F. Oshis, and M. V. Shimanskaya, “Conversion of heterocyclic compounds on membrane catalysts,” Khim. Geterotsikl. Soedin., 599–602 (1975).

  41. E. Dziluma, S. Giller (Hiller), S. Slavinskaya (Slavinska), V. Evgrashin, D. Kreile, A. Strautina, and J. Milman, “Some aspects of the genesis of vandium catalysts for vapor-phase oxidation and oxidative ammonolysis of heterocyclic and other compounds. Scientific bases for the preparation of heterogeneous catalysis.” An International Symposium, Brussels, 1975, B5, 1–10 (1975).

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  42. S. Giller (Hiller), A. Karmil'chik (Karmilchik), V. Stonkus, B. Kataev (Katayev), and M. Shimanskaya (Shymanska), Promoted chromium-zinc-manganese oxide catalyst for decarbonylation reactions and scientific principles of its preparation. An international Sympsoium, Brussels, 1975, F4, 1–8.

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VII. Physical Organic Chemistry

  1. G. Ya. Vanag, Ya. A. Éidus, and S. A. Giller, “Tautomerism and isomerism of 2-nitroindane-1,3-dione,” Dokl. Akad. Nauk SSSR, 79, 977–980 (1951).

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  2. Ya. P. Stradyn' and S. A. Giller, “Mechanism of the polarographic reduction of 2-nitrofuran,” Izv. Akad. Nauk LatvSSR, No. 10, 121–126 (1958).

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  3. Ya. P. Stradyn', S. A. Giller, and A. Ya. Dzene, “Polarographic reduction of some 5-nitrofuran derivatives used as chemotherapeutic agents,” Izv. Akad. Nauk LatvSSR, No. 12, 71–78 (1959).

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  4. Ya. P. Stradyn', S. A. Giller, and Yu. K. Yur'ev, “Polarographic reduction of 2-nitrofuran and 2-nitroselenophene derivatives,” Dokl. Akad. Nauk SSSR, 129, 816–819 (1959).

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  5. Ya. P. Stradyn, S. A. Giller, Yu. K. Yur'ev, and E. L. Zaitseva, “Polarographic study of 2-nitroselenophene derivatives,” Izv. Akad. Nauk LatvSSR, No. 3, 85–92 (1960).

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  6. Ya. P. Stradyn' and S. A. Giller, “Polarographic study of 5-substituted 2-nitrofuran derivatives,” Izv. Akad. Nauk LatvSSR, No. 2, 95–100 (1960).

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  7. Ya. A. Éidus, K. K. Venter, and S. A. Giller, “Effect of terminal substituents in 5- nitrofurylpolyene derivatives and their electronic spectra,” Dokl. Akad. Nauk SSSR, 141, 655–658 (1961).

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  8. I. B. Mazheika, S. A. Giller, P. A. Gembitskii, R. Ya. Levina, “Dipole moments of some phenylcyclopropane derivatives,” Zh. Obshch. Khim., 33, 1698–1699 (1963).

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  9. R. A. Gavar, Ya. P. Stradyn', and S. A. Giller, “Electrochemical generation of free-radical anions in a number of 5-nitrofuran derivatives,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 381 (1964).

  10. R. A. Gavar, Ya. P. Stradyn', and S. A. Giller, “Electrochemical generation of free-radical anions in the 5-nitrofuran series,” Dokl. Akad. Nauk SSSR, 157, 1424–1426 (1964).

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  11. R. A. Gavar, Ya. P. Stradyn', and S. A. Giller, “Recording of the ESR spectra of short-lived free-radical anions,” Zavod. Lab., 31, 41–45 (1965).

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  12. S. A. Giller, I. B. Mazheika, and I. I. Grandberg, “Electron density distribution in heterocyclic systems with two adjacent nitrogen atoms. II. Dipole moment of pyrazole,” Khim. Geterotsikl. Soedin., 103–106 (1965).

  13. S. A. Giller, I. B. Mazheika, and I. I. Grandberg, “Electron density distribution in heterocyclic systems with two adjacent nitrogen atoms. III. Dipole moments of some alkyl, aryl, and nitro derivatives of pyrazole,” Khim. Geterotsikl. Soedin., 107–111 (1965).

  14. A. Ya. Karmil'chik, S. A. Giller, and M. V. Shimanskaya, “Isotope exchange of furan with heavy water,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 328–331 (1966).

  15. J. Stradins, R. Gawars, G. Reihmanis, and S.Giller (Hillers), “Untersuchungen von intermediären Reduktionsprodukten der 2-Nitrofuran-Derivate mit Hilfe der Polarographie und der ESR Spektrometrie,” in: Electrochemische Methoden und Prinzipien in der Molekular Biologie. III Jenaer Symposium, 25 bis 29 Mai, 1965. Vorträge und Diskussionen. Berlin, 1966, pp. 601–610 (Abhandlungen der Deutschen Akademie der Wissenschaften zu Berlin. Klasse für Medizin, 1966, 4).

  16. I. B. Mazheika, G. I. Chipen, and S. A. Giller, “Electron density distribution in heterocyclic systems with two adjacent nitrogen atoms. IV. Dipole moments of some 1,2,4-triazole derivatives,” Khim. Geterotsikl. Soedin., 776–782 (1966).

  17. S. A. Giller, I. B. Mazheika, I. I. Grandberg, and L. I. Gorbacheva, “Electron density distribution in heterocyclic systems with two adjacent nitrogen atoms. V. Dipole moments of some halo, amino, and hydroxy derivatives of pyrazole,” Khim. Geterotsikl. Soedin., 130–134 (1967).

  18. S. A. Giller, I. B. Mazheika, and I. I. Grandberg, “Electron density distribution in heterocyclic systems with two adjacent nitrogen atoms. VI. Dipole moments of some bis-pyrazole systems and polycondensed systems containing a pyrazole ring,” Khim. Geterotsikl. Soedin., 884–888 (1967).

  19. Ya. A. Éidus, A. Ya. Ékmane, K. K. Venter, and S. A. Giller, Atlas of the Electronic Spectra of 5-Nitrofuran Compounds [in Russian], Zinatne, Riga (1968), p. 160.

  20. J. Éidus, A. Ya. Ekmane, K. K. Venters, and S. A. Giller (Hilier), Atlas of Electronic Spectra of 5-Nitrofuran Compounds, Ann Arbour Sci. Publishers, Inc., Portland, Oregon (1970).

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  21. K. K. Venter, Ya. A. Eidus, D. O. Lolya, and S. A. Giller, “Syntheses involving 5-nitro-2-furylpolyalkenals and 5-nitro-2-furylpolyalkenones. VIII. Synthesis and electronic and vibrational spectra of some ω,ω′-bis-(5-nitro-2-furyl)polyalkenes,” Khim. Geterotsikl. Soedin., 405–412 (1968).

  22. Ya. P. Stradyn', R. A. Gavar, V.K. Grin', and S. A. Giller, “Stability and kinetics of the disappearance of anion radicals of the nitrofuran series,” Teor. Eksp. Khim. (Kiev), No. 4, 774–779 (1968).

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  23. M. G. Voronkov, S. A. Giller, I. N. Goncharova, L. I. Mironova, and V. P. Feshin, “Cl35 Nuclear quadrupole resonance of alkane-α,ω-dicarboxylic acid chlorides,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 250–251 (1969).

  24. G. P. Sokolov and S. A. Giller, “Synthesis of cyclic diacetals of fumaraldehyde, α,α′-dibromosuccinaldehyde, and 2-butynedial,” Khim. Geterotsikl. Soedin., 32–35 (1969).

  25. R. A. Gavar, V. A. Zilitis, Ya. P. Stradyn', and S. A. Giller, “π-Electron structure of the nitrofuran system. I. Distribution of the unpaired electron in anion radicals of 5-nitrofuran and its 2-substituted derivatives,” Khim. Geterotsikl. Soedin., 294–298 (1970).

  26. R. A. Gavar, V. A. Zilitis, Ya. P. Stradyn', and S. A. Giller, “π-Electron structure of the nitrofuran system. II. Molecular orbitals of the π electrons of 5-nitrofuran and its 2-substituted derivatives,” Khim. Geterotsikl, Soedin., 3–8 (1971).

  27. A. D. Garnovskii, Yu. V. Kolodyazhnyi, O. A. Osipov, V. I. Minkin, S. A. Giller, I. B. Mazheika, and I. I. Grandberg, “Dipole moments and structures of azoles,” Khim. Geterotsikl. Soedin., 867–892 (1971).

  28. G. O. Reikhmanis, Ya. P. Stradyn', R. A. Gavar, and S. A. Giller, “Electrochemical and protolytic transformations of α-phenyl- and α-(2-furyl)-β-nitroethylene,” Zh. Obshch. Khim., 41, 906–910 (1971).

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  29. I. K. Tutane, Ya. P. Stradyn', B. V. Kurgan, and S. A. Giller., “Polarographic behavior of thiol ethers of aromatic and furan carboxylic acids,” Zh. Obshch. Khim., 41, 1912–1915 (1971).

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  30. Ya. P. Stradyn', I. Ya. Kravis, G. O. Reikhmanis, and S. A. Giller, “Polarographic study of the conductivity of the polar effect of a substituent through the furan ring and side bridged groupings,” Khim. Geterotsikl. Soedin., 1309–1312 (1972).

  31. R. A. Gavar, L. Kh. Baumane, Ya. P. Stradyn', and S. A. Giller, “π-Electron structure of the nitrofuran system. III. Effect of the medium on the character of the ESR spectra of anion radicals of 5-nitrofurans,” Khim. Geterotsikl. Soedin., 435–440 (1972).

  32. I. V. Turovskii, V. T. Glezer, L. Ya. Avota, Ya. P. Stradyn', and S. A. Giller, “Protolysis constants of 6-pyridazone derivatives,” Khim. Geterotsikl. Soedin., 993–995 (1973).

  33. Ya. P. Stradyn', V. P. Kadysh, and S. A. Giller, “Polarography of heterocyclic compounds. I. General data on the polarographic behavior of heterocycles and electrochemical reduction of heteroaromatic compounds,” Khim. Geterotsikl. Soedin., 1587–1603 (1973).

  34. V. T. Glezer, Ya. P. Stradyn', I. K. Tutane, L. Ya. Avota, and S. A. Giller, “Polarographic reduction of 6-pyridazone and its derivatives,” Zh. Obshch. Khim., 43, 1150–1153 (1973).

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  35. G. P. Sokolov and S. A. Giller, “Stereochemistry of bisdioxolane systems. I. Synthesis and configuration of isomers of 1,2-bis [4-(p-tosyloxymethyl)-1,3-dioxolan-2-yl]ethane,” Khim. Geterotsikl. Soedin., 1608–1610 (1973).

  36. R. A. Gavar, L. Kh. Baumane, Ya. P. Stradyn', and S. A. Giller, “π-Electron structure of the nitrofuran system. IV. ESR Spectra of the anion radicals of 2-vinylene derivatives of 5-nitrofuran,” Khim. Geterotsikl. Soedin., 324–329 (1974).

  37. B. V. Kurgane, A. K. Grinvalde, Ya. P. Stradyn', M. T. Brakmane, and S. A. Giller, “Enolizability of thiol esters of acetoacetic and malonic acids,” Zh. Organ. Khim., 11, 2306–2309 (1974).

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  38. Ya. P. Stradyn', V. P. Kadysh, and S. A. Giller, “Polarography of heterocyclic compounds. II. Heteroethylene and heteroparaffin compounds. Effect of substituents in the side chain on the parameters of electrical reduction of heterocyclic compounds,” Khim. Geterotsikl. Soedin., 147–162 (1974).

  39. V. A. Pestunovich, V. G. Sidorkin, V. A. Shagun, M. G. Voronkov, S. A. Giller, É. É. Liepin'sh, and A. V. Eremeev, “Conformational analysis of 2-phenyl-1, 3-diazabicyclo [3.1.-0]hexane,” Khim. Geterotsikl. Soedin., 936–940 (1975).

  40. S. A. Giller, É. É. Liepin'sh, A. V. Eremeev, and V. A. Kholodnikov, “PMR spectra of 1,3-diazabicyclo[3.1.0] hexanes in the presence of tris (dipivaloylmethanato) europium,” Khim. Geterotsikl. Soedin., 940–942 (1975).

VIII. Organic Analysis

  1. Ya. P. Stradyn', S. A. Giller, and L. K. Lepin', “Determination of the solubility of nitrofurans in water by means of polarography,” Izv. Akad. Nauk LatvSSR, No. 1, 113–120 (1958).

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  2. S. A. Giller, A. Ya. Krauya, and Z. Ya. Zelmene, “Method for the quantitative determination of mercury in mercuirichlorides of the furan series,” Izv. Akad. Nauk LatvSSR, No. 4, 75–79 (1959).

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  3. M. V. Shiraanskaya, S. A. Giller, and V. A. Slavinskaya “Standardization of the quality of industrial-grade furfural,” Khim. Prom. (Riga), No. 2, 20–22 (1961).

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  4. V. É. Égert, M. V. Shimanskaya, and S. A. Giller, “Methods for the quantitative determination of 5-nitrofurans. I. Modified Kjeldahl method for the determination of 5-nitrofurfural derivatives, Izv. Akad. Nauk LatvSSR, Ser. Khim., 55–60 (1961).

  5. V. É. Égert, M. V. Shimanskaya, and S. A. Giller, “Methods for the quantitative determination of 5-nitrofurans. III. Colorimetry,” Akad. Nauk LatvSSR, Ser. Khim., 199–204 (1961).

  6. S. A. Giller, V. É. Égert, and M. V. Shimanskaya, “Analytical determination of furazolidone,” in: Furazolidone [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1962), pp. 17–27.

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  7. V. É. Égert, M. V. Shimanskaya, and S. A. Giller, “Methods for the quantitative determination of 5-nitrofurans. IV. Potentiometric determination of N-(5′-nitro-2′-furfurylidene)-1-aminohydantoin (furadonine),” Izv. Akad. Nauk LatvSSR, Ser. Khim., 39–43 (1962).

  8. S. A. Giller, V. É. Égert, M. V. Shimanskaya, and S. K. Germane, “Methods for the quantitative determination of 5-nitrofurans. V. Spectrophotometeric determination on N-(5′-nitro-2′-furfurylidene)-3-amino-2-oxazolidone (furazolidone) in the presence of some impurities,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 577–581 (1962).

  9. A. A. Anderson, A. Ya. Karmil'chik, M. V. Shimanskaya, and S. A. Giller, “Application of gas—liquid chromatography for the analysis of furan and its derivatives,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 168–176 (1963).

  10. Ya. P. Stradyn', I. F. Aizpuriete, and S. A. Giller, “Polarographic study of a new antibacterial preparation — furazoline,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 29–34 (1963).

  11. Ya. P. Stradyn', I. K. Tutane, M. A. Alberta, and S. A. Giller, “Polarographic behavior of furothiazole [2-acetamido-4-(5-nitro-2-furyl)-thiazole],” Izv. Akad. Nauk LatvSSR, Ser. Khim., 371–376 (1963).

  12. V. É. Égert, M. V. Shimanskaya, and S. A. Giller, “Methods for the quantitative determination of 5-nitrofurans. VI. Conductometric determination of 5-nitrofuran derivatives containing a hydantoin ring (furadonine and furazidine),” Izv. Akad. Nauk LatvSSR, Ser. Khim., 177–180 (1963).

  13. V. É. Égert, S. A. Giller, A. A. Lielgalve, and M. V. Shimanskaya, “Methods for the quantitative determination of 5-nitrofurans. VII. Spectrophotometric determination,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 531–540 (1963).

  14. A. A. Anderson, A. Ya. Karmil'chik, M. V. Shimanskaya, and S. A. Giller, “Application of gas-liquid chromatography for the analysis of mixtures of furan compounds,” in: Molecular Chromatography [in Russian], Izd. Akad. Nauk SSSR, Moscow (1964), pp. 52–57.

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  15. A. Ya. Karmil'chik, V. V. Stonkus, M. V. Shimanskaya, and S. A. Giller, “Chromatographic analysis of furfural,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 543–546 (1967).

  16. S. A. Giller, V. É. Égert, M. V. Shimanskaya, and Ya. P. Stradyn', “Analytical determination of furagin and solafur,” in: Furagin and Solafur [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1968), pp. 7–31.

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  17. A. Ya. Karmil'chik, V. V. Stonkus, L. S. Efimova, M. V. Shimanskaya, and S. A. Giller, “Chromatographic analysis of mixtures containing methylfurfural,” Izv. Akad. Nauk Latv-SSR, Ser. Khim., 29–32 (1968).

  18. S. A. Giller, V. É. Égert, K. K. Venter, N. Ya. Ozolinya, A. A. Lielgalve, and D. O. Lolya, “Analytical determination of maleic acid hydrazide and its salts,” in: Maleic Acid Hydrazide as a Plant-Growth Regulator [in Russian], Nauka, Moscow (1973), pp. 310–318 (1973).

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  19. A. A. Avots, V. D. Shatts, and A. Ya. Karmil'chik, “Study of the hydrogenolysis of furan derivatives by means of pulse chromatography,” in: Chromatographic Analysis in Wood Chemistry [in Russian], Zinatne, Riga (1975), pp. 162–168.

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IX. Interrelationship between Structure and Physiological Activity

  1. S. A. Giller, “Possible reason for the bacterial activity of some organic compounds, particularly derivatives of the furan series,” Izv. Akad. Nauk LatvSSR, No. 12, 15–44 (1948).

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  2. K. K. Medne, S. A. Giller, S. K. Germane, and K. K. Venter, “Interrelationship between chemical structure and the antituberculous activity of some compounds of the 5-nitrofuran series,” in: Problems of Tuberculosis [in Russian], Vol. 7, Chemotherapy [in Russian], Riga (1967), pp. 373–380.

  3. J. Stradin'sh (Stradins), S. Giller (Hiller), R. Gavars, G. Reikhmanis (Reihmanis), and L. Baumane, “Electrochemical properties and biological activity of nitrofurans,” in: Biological Aspects of Electrochemistry. Proceedings of the First International Symposium, May 31 to June 4, 1971, Basel-Stuttgart (1971), pp. 607–617.

  4. S. A. Giller, A. B. Glaz, V. E. Golender, L. A. Rastrigin, and A. B. Rozenblit, “Application of the theory of sample recognition for the prediction of the pharmacological activity of chemical compounds,” Khim.-Farmats. Zh., No. 12, 18–22 (1972).

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  5. S. A. Giller, V. E. Golender, A. B. Rosenblit, L. A. Rastrigin, and A. B. Glaz, “Cybernetic methods of drug design. I. Statement of the problem — the perceptron approach,” Computers and Biomed. Res., No. 6, 411–414 (1973).

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X. Search for and Study of Antibacterial and Antituberculous Substances

  1. S. A. Giller, “Research of the Academy of Sciences of the Latvian SSR on the industrial incorporation and medical adoption of new medicinal preparations [synthesis and production of the antituberculous preparation PASK],” Izv. Akad. Nauk LatvSSR, No. 12, 27–46 (1950).

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  2. S. A. Giller, A. K. Lokenbakh, and L. A. Mai, “Research on the synthesis of 4-aminosalicylic acid,” in: p-Aminosalicylic Acid (PASK) in Tuberculosis Therapy [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1950), pp. 7–25.

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  3. S. A, Giller, M. Yu. Lidak, M. Ya. Berklava, and M. V. Tarvid, “Antituberculous activity of a preparation containing isonicotinoylhydrazide,” Izv. Akad. Nauk LatvSSR, No. 10, 157–160 (1952).

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  4. S. A. Giller, M. Yu. Lidak, M. Ya. Berklava, and M. V. Tarvid, “Antituberculous activity of a preparation containing isonicotinoylhydrazide,” in: Tubazid [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1968).

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  5. S. A. Giller, Ya. P. Stradyn', and N. S. Ratenberg, “Dynamics of the excretion of some new preparations of the nitrofuran series from the organism,” Izv. Akad. Nauk LatvSSR, No. 3, 107–114 (1959).

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  6. S. P. Zaeva, S. A. Giller, S. K. Germane, Ya. P. Stradyn', L. N. Alekseeva, L. V. Kruzmetra, M. A. Alberta, I. F. Aizpuriete, and R. Yu. Kalnberg, “Experimental study of a new preparation of the nitrofuran series — furazoline (F-150),” Zh. Mikrobiol. Epidemiol, i Immunobiol., No. 10, 17–20 (1961).

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  7. S. A. Giller and R. Yu. Kalnberg, “Synthesis of furazolidone,” in: Furazolidone [in Russian], Izd. Akad. Nauk LatvSSR, Riga, 5–15 (1962).

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  8. S. A. Giller, K. K. Medne, K. K. Venter, S. K. Germane, and A. Ya. Zile, “Study of the tuberculostatic activity of some derivatives of unsaturated aldehydes and ketones of the 5-nitrofuran series,” Dokl. Akad. Nauk SSSR, 144, 108–111 (1962).

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  9. S. A. Giller, S. P. Zaeva, K. K. Venter, L. N. Alekseeva, L. V. Kruzmetra, and S. K. Germane, “Syntheses involving 5-nitro-2-furylpolyalkenals and 5-nitro-2-furylpolyalkenones. VII. Synthesis and study of the antibacterial properties of derivatives of α,β-unsaturated and polyene aldehydes and ketones of the 5-nitrofuran series,” Khim. Geterotsikl. Soedin., 187–194 (1965).

  10. S. A. Giller, A. Ya. Zile, L. V. Kruzmetra, V. I. Vereshchagina, K. K. Venter, and S. P. Korshunov, “Antibiotic activity of some acetylenic derivatives of furan,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 104–108 (1967).

  11. R. Yu. Kalnberg, K. K. Venter, B. A. Brizga, L. N. Alekseeva, L. V. Kruzmetra, and S. A. Giller, “Synthesis and antibacterial properties of some 5-morpholinomethyl-3-amino-2- oxazolidone derivatives of the 5-nitrofuran series,” Khim.-Farmats. Zh., No. 11, 47–49 (1967).

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  12. S. P. Zaeva, S. A. Giller, M. V. Shimanskaya, V. É. Égert, K. K. Venter, L. V. Kruzmetra, M. A. Alberta, L. N. Alekseeva, S. K. Germane, E. K. Brentsis, F. N. Branover, B. O. Press, and G. A. Grigalinovich, “Experimental study of a new chemotherapeutic preparation — solafur,” in: Furagin and Solafur [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1968), pp. 33–40.

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  13. S. A. Giller, K. K. Medne, and R. Yu. Frim, “Tuberculostatic action of some derivatives of 5-(p-, m-, and o-nitrophenyl)furfurals,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 133–136 (1969).

  14. N. O. Saldabol, L. N. Alekseeva, B. A. Brizga, L. V. Kruzmetra, and S. A. Giller, “Synthesis and antimicrobial action of furyl-substituted indolizines, imidazo [1,2-a]pyrimidines, and imidazo [1,1-b] thiazoles,” Khim.-Farmats. Zh., No. 7, 20–25 (1970).

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  15. A. F. Blyuger, S. A. Giller, M. K. Indulen, É. N. Kibitkina, É. Z. Krupnikova, Ya. Yu. Polis, E. P. Semushina, and P. P. Khvatov, “Study of the chemoprophylaxis of influenza by means of aminoadamantane derivatives,” in: Chemoprophylaxis and Chemotherapy of Influenza [in Russian], Leningrad (1972), pp. 142–145.

  16. S. A. Giller, L. A. Vol'f, and A. L. Meos, “Method for the modification of films and fibers in order to impart antibacterial properties to them,” French Patent No. 1368858 (1964).

  17. S. A. Giller, L. A. Vol'f, and A. I. Meos, “Method for the imparting of antibacterial properties to articles obtained from polyvinyl alcohol,” US Patent No. 3390008 (1968).

  18. S. A. Giller, V. V. Kotetskii, Ya. A. Kharit, L. A. Vol'f, and K. K. Venter, “Chemical fiber having antibacterial properties,” British Patent No. 1254702 (1972).

XI. Study of Fungicidal Preparations

  1. S. A. Giller, A. Ya. Zile, and M. Ya. Berklava, “Method for the treatment of skin diseases. The preparation nitrofurylene,” USSR Author's Certificate No. 186635; Byul. Izobr., No. 19, 70 (1966).

  2. S. A. Giller, M. A. Alberta, A. Ya. Zile, L. I. Vereshchagin, K. K. Venter, and S. P. Korshunov, “Fungistatic activity of some acetylenic derivatives of furan and their effect on the respiratory intensity and the catalase activity of pathogenic fungi,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 63–68 (1966).

  3. N. O. Saldabol, S. A. Giller, L. N. Alekseeva, and B. A. Brizga, “Syntheses in the methyl 2-furyl ketone series. XII. (5-Nitro-2-furyl)-substituted imidazoheterocyclic compounds with a nitrogen atom in common,” Khim.-Farmats. Zh., No. 2, 27–31 (1967).

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  4. S. A. Giller, A. Ya. Zile, M. Ya. Berklava, B. O. Press, and K. K. Medne, “Fungistatic activity of some alcohols and esters of the nitrofuran series,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 121–124 (1969).

  5. S. A. Giller, A. Ya. Zile, M. Ya. Berklava, L. V. Kruzmetra, S. K. Germane, B. O. Press, M. A. Alberta, and G. A. Grigalinovich, “Nitrofurylene — A new original Soviet fungistat,” in: Experimental and Clinical Pharmacotherapy [in Russian], Vol. 1, Riga (1970), pp. 111–121.

XII. Study of Antiblastic Properties

  1. M. Yu. Lidak, S. A. Giller, and A. Ya. Medne, “Synthesis of some bifunctional derivatives of ethyleneimine with antiblastic action,” Izv. Akad. Nauk LatvSSR, No. 1, 87–90 (1959).

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  2. M. Yu. Lidak, S. A. Giller, and A. Ya. Medne, “Synthesis of ThioTEFA,” in: ThioTEFA [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1961), pp. 5–8.

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  3. M. Yu. Lidak and S. A. Giller, “New ethyleneimine-containing cancerolytic polymers. New cancerostatic derivatives of ethyleneimine. Study of the reaction of ethyleneimine with derivatives containing carbonyl and carboxyl functions,” in: Methods for the Synthesis of and Search for Antitumorigenic Preparations, [in Russian], Izd. Akad. Med. Nauk SSSR, Moscow (1962), pp. 150–156.

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  4. S. A. Giller, M. Yu. Lidak, R. K. Bane, and I. Ya. Birkmane, “Synthesis and technology of cyclophosphane,” in: Cyclophosphane [in Russian], Izd. Akad. Nauk LatvSSR, Riga (1965), PP. 7–12.

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  5. S. A. Giller, M. Yu. Lidak, A. A, Zidermane, and A. G, Pinus, “Method for the treatment of erythremia. The preparation ‘imifos’,” USSR Author's Certificate No. 182877; Byul. Izobr., No. 12, 82 (1966).

  6. S. A. Giller, M. Yu. Lidak, and E. Ya. Markava, “Synthesis of new phosphoramides and thiophosphoramides for the treatment of malignant tumors,” in: Imifos [in Russian], Izd. Akad. Nauk. LatvSSR, Riga (1968), pp. 11–23.

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  7. R. Yu. Kalnberg, K. K. Venter, N. M. Sukhova, A. A. Zidermane, A. Zh. Dauvarte, M. Yu. Lidak, and S. A. Giller, “Synthesis and study of the cytotoxic properties of bis(2-chlorethyl)amino and N,N-bis(2-chloroethyl)hydrazino derivatives,” Khim.-Farmats. Zh., No. 2, 10–16 (1968).

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  8. R. Yu. Kalnberg, S. A. Giller, M. Yu. Lidak, L. N. Alekseeva, L. V. Kruzmetra, B. A. Brizga, A. Ya. Zile, and I. O. Petersone, “Synthesis and study of the biological activity of methyldithiocarbazonates of unsaturated aldehydes of the 5-nitrofuran series,” Khim.-Farmats. Zh., No. 11, 11–13 (1968).

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  9. S. A. Giller, M. Yu. Lidak, K. K. Venter, R. Yu. Kalnberg, A. A. Ziderman, A. Zh. Dauvarte, and N. M. Sukhova, “Method for the preparation of N,N-[β-(5′-nitro-2′-furyl)-alkylidene]bis(2-chloroethyl) hydrazone(nifurone),” USSR Author's Certificate No. 257508; Byul. Izobr., No. 36, 29 (1969).

  10. S. A. Giller, M. Yu. Lidak, N. M. Sukhova, and K. K. Venter, “Method for the preparation of 2-[2′-(5′'-nitro-2′'-furyl) butadienyl]quinoline derivatives,” USSR Author's Certificate No. 242174; Byul. Izobr., No. 15, 26 (1969).

  11. S. A. Giller, M. Yu. Lidak, N. M. Sukhova, A. V. Eremeev, A. A. Ziderman, and I. I. Sablina, “Method for the preparation of substituted hydrazones of 4-carboxy-2-formylquinoline derivatives,” USSR Author's Certificate No. 333168; Byul. Izobr., No. 11, 97 (1972).

  12. A. Zh. Dauvarte, A. A. Ziderman, R. Yu. Kalnberga, M. Yu. Lidak, K. K. Venter, N. M. Sukhova, R. K. Verpele, and S. A. Giller, “Antitumorigenic activity of some derivatives of the 5-nitrofuran series,” in: Antitumorigenic Compounds of the 5-Nitrofuran Series. Experimental Studies [in Russian], Zinatne, Riga (1972), pp. 17–24.

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  13. R. Yu. Kalnberga, S. A. Giller, M. Yu. Lidak, and N. M. Sukhova, “Synthesis of bis (2- chloroethyl)hydrazino and bis (2-chloroethyl)amino derivatives of 5-nitrofuran,” in: Antitumorigenic Compounds of the 5-Nitrofuran Series. Experimental Studies [in Russian], Zinatne, Riga (1972), pp. 31–32.

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  14. A. Zh. Dauvarte, A. A. Zidermane, R. Yu. Kalnberga, M. Yu. Lidak, B. V. Kurgane, N. M. Sukhova, and S. A. Giller, “Antitumorigenic activity of N,N-bis(2-chloroethyl)hydrazino derivatives of aromatic and heterocyclic aldehydes,” in: Antitumorigenic Compounds of the 5-Nitrofuran Series. Experimental Studies [in Russian], Zinatne, Riga (1972), pp. 33–37.

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  15. S. A. Giller, R. A. Zhuk, M. Yu. Lidak, and A. A. Ziderman, “New antitumorigenic preparations based on uracil derivatives,” Belgian Patent No. 708903 (1968).

  16. S. A. Giller, M. Yu. Lidak, K. K. Venter, R. Yu. Kalnberg, A. A. Ziderman, and A. Zh. Dauvarte, “Method for the preparation of N,N-bis (2-chlorethyl)hydrazones of the 5-nitrofuran series,” French Patent No. 154094 (1968); US Patent No. 1137467 (1968); French Patent No. 7161M (1969); Japanese Patent No. 577404 (1970); US Patent No. 3526643 (1970).

  17. S. A. Giller, R. A. Zhuk, M. Yu. Lidak, and A. A. Ziderman, “New method for the preparation of uracil derivatives,” French Patent No. 1574684 (1969); British Patent No. 1168391 (1969); French Patent No. 7448M (1969).

  18. S. A. Giller, M. Yu. Lidak, É. M. Markava, and A. A. Ziderman, “Phosphorus-containing derivatives of diethyleneimide,” British Patent No. 1052711 (1967).

  19. S. A. Giller, M. Yu. Lidak, É. M. Markava, and A. A. Ziderman, “Method for the preparation of diethyleneimides of phosphoric and thiophosphoric acids,” Japanese Patent No. 552461 (1968); West German Patent No. 1285475 (1968); Swiss Patent No. 319771 (1970).

  20. S. A. Giller, R. A. Zhuk, M. Yu. Lidak, and A. A. Ziderman, “Method for the preparation of N1-(2′-tetrahydrofuryl) and N1-(2′-tetrahydropyranyl) derivatives of 5-substituted uracils and their alkali-metal salts,” Swiss Patent No. 493557 (1970).

  21. S. A. Giller, M. Yu. Lidak, A. Zh. Dauvarte, R. Yu. Kalnberga, A. A. Stengrevich, V. A. Klyavinya, A. A. Zidermane, and O. I. Starkova, “Method for the preparation of β-bis(2-chlorethyl)hydrazones,” USSR Author's Certificate No. 445275; Byul. Izobr., No. 33, 184 (1975).

  22. A. A. Lazdyn'sh, D. Ya. Sniker, A. K. Veinberg, S. A. Giller, I. L. Knunyants, L. S. German, and V. A. Kozmina, “Method for the preparation of 5-fluorouracil,” British Patent No. 1323785 (1973); US Patent No. 3846429 (1974).

  23. S. A. Giller, R. A. Zhuk, A. É. Berzin', L. A. Sherin', and A. A. Lazdyn'sh, “Method for the preparation of N1-(2′-furanidyl) derivatives of 5-substituted uracils,” Belgian Patent No. 807556 (1974).

XIII. Study of Neurotropic and Psychotropic Compounds

  1. S. A. Giller, Kh. M. Vasserman, and K. K. Venter, “Synthesis of some new ganglion-blocking and curarelike substances from furfural,” in: Problems in the Utilization of Pentosan-Containing Raw Material [in Russian], Riga (1958), pp. 393–401.

  2. S. A. Giller, G. P. Sokolov, V. E. Klusha, and A. A. Kimenis, “Method for the preparation of 1,2-bis(4′-pyrrolidinomethyl-1,3′-dioxolan-2′-yl)ethane dimethiodide (dioxonium),” USSR Author's Certificate No. 267634; Byul. Izobr., No. 4, 13 (1959).

  3. Kh. M. Vasserman and S. A. Giller, “Utilization of saturated nitrogen-containing heterocycles for the synthesis of ganglion-blocking and curarelike substances,” in: Chemistry, Technology, and Application of Pyridine and Quinoline Derivatives [in Russian], Riga (1960), pp. 207–221.

  4. S. A. Giller, É. A. Baumanis, G. P. Sokolov, and V. Ya. Grinshtein, “Synthesis and Anti-MAO Activity of Alkylhydrazides of Pyridazine-3-carboxylic Acid,” Dokl. Akad. Nauk SSSR, 145, 440–442 (1962).

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  5. G. P. Sokolov, and S. A. Giller, “Method for the preparation of quaternary salts of 1,2-bis(4′-R,R-aminomethyl-1′,3′-dioxolan-2′-yl)ethane,” USSR Author's Certificate No. 196883; Byul. Izobr., No. 12, 42 (1967).

  6. G. P. Sokolov, V. E. Klusha, A. A. Kimenis, and S. A. Giller, “Synthesis and curarizing action of quaternary salts of bisaminomethyldioxolanylethane and bisaminomethyldioxolanyl ethylene,” Khim.-Farmats Zh., No. 3, 3–7 (1968).

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  7. G. P. Sokolov, S. A. Giller, A. A. Kimenis, V. E. Klusha, and Ya. Ya. Ginters, “Medicinal agent,” USSR Author's Certificate No. 278963; Byul. Izobr., No. 26, 82 (1970).

  8. G. P. Sokolov, A. A. Kimenis, D. K. Kruskop, V. E. Klusha, and S. A. Giller, “Synthesis and pharmacological properties of cyclic diacetals of sebacaldehyde,” Khim.-Farmats. Zh., No. 2, 10–14 (1972).

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  9. G. P. Sokolov, R. O. Vitolin', and S. A. Giller, “Synthesis and pharmacological properties of the hydrochlorides and methiodides of aminomethyl derivatives of 2-[diphenyl (hydroxy)methyl]-1,3-dioxolane,” Khim.-Farmats Zh., No. 12, 10–15 (1973).

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  10. G. P. Sokolov, S. A. Giller, A. A. Kimenis, V. E. Klusha, Ya. Ya. Ginters, and M. M. Veveris, “Dioxonium — a new curarelike agent,” Khim.-Farmats. Zh., No. 2, 60–61 (1974).

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  11. G. P. Sokolov, A. A. Kimenis, M. M. Veveris, and S. A. Giller, “Synthesis and curarelike properties of quaternary ammonium derivatives of cyclic acetals of levulinaldehyde and levulinic acid,” Khim.-Farmats. Zh., No. 3, 8–13 (1973).

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  12. S. A. Giller, G. P. Sokolov, A. A. Kimenis, and V. E. Klusha, “Method for the preparation of 1,2-bis(4′-pyrrolidinomethyl-1′,3′-dioxolan-2′-yl) ethane,” Belgian Patent No. 743137 (1970); US Patent No. 3661929 (1972); Japanest Patent No. 26787 (1972); French Patent No. 2059981 (1973); West German Patent No. 1923843 (1974).

  13. S. A. Giller, G. P. Sokolov, A. A. Kimenis, and V. E. Klusha, “Method for the preparation of 1,2-bis(4′-pyrrolidinomethyl-1′, 3′-dioxolan-2′-yl)ethane dimethiodide,” Swiss Patent No. 503049 (1971).

  14. S. A. Giller, G. P. Sokolov, A. A. Kimenis, and V. E. Klusha, “Changes in natural dioxolane derivatives and their utilization for pharmaceutical preparations,” British Patent No. 1244437 (1971).

XIV. Technology of the Manufacture of Organic Compounds

  1. S. A. Giller, M. V. Shimanskaya, and I. I. Ioffe, “Vapor-phase catalytic oxidation of furfural to maleic anhydride,” in: Problems in the Utilization of Pentosan-Containing Raw Material [in Russian], Riga (1958), pp. 263–275.

  2. M. M. Gershov and S. A. Giller, “Method for the purification of technical-grade p-aminosalicylic acid,” USSR Author's Certificate No. 118212; Byul. Izobr., No. 19, 33 (1959).

  3. S. A. Giller, É. V. Zarin'sh, and M. M. Gershov, “Method for the preparation of p-amino-salicyclic acid by carbonation of m-aminophenol,” USSR Author's Certificate No. 118213; Byul. Izobr., No. 4, 13 (1959).

  4. M. V. Shimanskaya and S. A. Giller, “Development of a new method for the industrial production of maleic anhydride,” Khim. Prom., No. 3, 25–28 (1960).

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  5. M. V. Shimanskaya and S. A. Giller, “Preparation of synthetic pyruvic and malic acids from inedible raw material,” in: Material from the Scientific-Technical Conference on the Intensification of Processes for the Manufacture of Nutritive Acids [in Russian], Riga (1961), pp. 113–122.

  6. A. A. Avot, M. V. Shimanskaya, S. A. Giller, V. A. Slavinskaya, M. K. Sile, and I. Ya. Silis, “Pilot apparatus for the study of catalytic vapor-phase oxidation processes,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 209–215 (1967).

  7. A. Ya. Karmil'chik, V. V. Stonkus, M. V. Shimanskaya, and S. A. Giller, “Industrial method for the preparation of α-methylfuran,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 747–748 (1969).

  8. S. A. Giller, A. Ya. Karmil'chik, A. A. Avot, A. P. Zeibot, V. A. Kupleniek, G. A. Énin'sh, V. V. Stonkus, M. V. Shimanskaya, “New technology for the preparation of furan,” Gidrolizn. Lesokhim. Prom., No. 4, 9–11 (1970).

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  9. A. Ya. Karmil'chik, V. V. Stonkus, M. V. Shimanskaya, and S. A. Giller, “Preparation of α-methylfuran from still residues from furfural production,” Gidrolizn. Lesokhim. Promysh., No. 7, 12–14 (1970).

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  10. Zh. É. Musha, S. A. Giller, and M. V. Shimanskaya, “Dehydration of Maleic Acid. III. Periodic dehydration with an experimental industrial apparatus,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 182–190 (1970).

  11. Zh. É. Musha, S. A. Giller, M. V. Shimanskaya, R. A. Liepinya, and Ya. P. Zile, “Desublimation of maleic anhydride from the contact gases from the oxidation of furfural,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 175–181 (1970).

  12. B. O. Polishchuk, V. V. Kotetskii, E. I. Shapiro, L. A. Vol'f, and S. A. Giller, “Preparation of an antimicrobial acetate fiber for medical purposes,” Khimicheskie Volokna, No. 4, 64–65 (1970).

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  13. A. A. Anderson, S. P. Yurel', M. V. Shimanskaya, and S. A. Giller, “Monitoring of the production of piperazine,” in: Gas Chromatography. A Collection of Scientific Works [in Russian], Moscow (1971), pp. 61–64.

  14. Zh. É. Musha, S. A. Giller, Ya. P. Zile, and M. V. Shimanskaya, “Rectification of maleic anhydride with an experimental industrial apparatus,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 59–63 (1971).

  15. Zh. É. Musha, S. A. Giller, M. V. Shimanskaya, and Ya. P. Zile, “Search for methods for the preservation of the colorlessness of commercial-grade maleic anhydride on prolonged storage,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 356–364 (1971).

  16. S. A. Giller, K. K. Venter, V. A. Kuplenieks, G. D. Tirzit, Kh. I. Girshovich, Z. G. Fridman, and S. G. Fridlender, “Synthesis and technology of the manufacture of the maleic acid hydrazide preparations GMK-T and GMK-Na,” in: Maleic Acid Hydrazide as a Plant-Growth Regulator [in Russian], Nauka, Moscow (1973), pp. 343–350.

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  17. S. A. Giller, K. K. Venter, A. A. Lazdyn'sh, R. Yu. Kalnberga, D. O. Lolya, V. V. Tsirule, V. É. Égert, and V. K. Ulaste, “Synthesis of β-(5-nitro-2-furyl) acrolein and optimization of the processes used to prepare it,” Khim.-Farmats. Zh., No. 2, 29–33 (1974).

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  18. A. A. Avots, A. Ya. Karmil'chik, V. V. Stonkus, V. S. Aizbalt-s, M. V. Shimanskaya, and S. A. Giller, “Technology for the preparation of α-methylfuran from methylfurfural,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 233–238 (1975).

XV. History and Organization of Science

  1. S. A. Giller, “The life and work of [Professor and Doctor of Chemical Sciences] Paul Kalnin',” Izv. Akad. Nauk LatvSSR, No. 12, 155–160 (1956).

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  2. A. I. Kalnin'sh and S. A. Giller, “Possibility of the utilization of woodcutting waste products,” in: Status and Prospects for the Study of the Plant Resources of the USSR [in Russian], Izd. Akad. Nauk. SSSR, Moscow-Leningrad (1958), pp. 204–212.

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  3. S. A. Giller, “Advances in organic synthesis. Research of the Institute of Organic Synthesis of the Academy of Sciences of the Latvian SSR,” Izv. Akad. Nauk LatvSSR, No. 4, 24–33 (1966).

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  4. S. A. Giller, “Corresponding Member of the Academy of Sciences of the Latvian SSR Mikhail Grigor'evich Voronkov,” Izv. Akad. Nauk LatvSSR, No. 4, 138–139 (1966).

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  5. S. A. Giller and A. R. Val'dman, “Yan Voldemarovich Peive [on his 60th birthday],” Izv. Akad. Nauk LatvSSR, No. 7, 149–151 (1966).

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  6. S. A. Giller, “Prospects for the development of scientific research in 1971–1975 in the institutes of the division of chemical and biological sciences of the Academy of Sciences of the Latvian SSR,” Izv. Akad. Nauk LatvSSR, No. 3, 22–31 (1968).

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  7. S. A. Giller, “Results of the most important scientific research in the chemical and biological sciences and their application in the national economy,” Izv. Akad. Nauk LatvSSR, No. 3, 19–24 (1969).

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  8. S. A. Giller, “Bioorganic chemistry and technical progress,” Izv. Akad. Nauk LatvSSR, No. 3, 90–98 (1970).

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  9. S. A. Giller, “Results of the most important scientific research in the chemical and biological sciences and their application in the national economy,” Izv. Akad. Nauk LatvSSR, No. 3, 20–28 (1970).

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  10. S. A. Giller, “From the history of the establishment and development of the scientific activity of the Institute of Organic Synthesis,” Izv. Akad. Nauk LatvSSR, No. 3, 80–87 (1971).

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XVI. Other Research

  1. P. Kalnins and S. Giller (Hillers), Par α-laktonu pastavesanas iespeju (1. zinojums par kada spilgts krasaina dimera ketena strukturus),” LatvPSR ZA Vestis, No. 2, 171–184 (1947); “The existence of α-lactones (first communication regarding the structute of an intensely colored ketene dimer).”

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  2. G. Ya. Vanag, S. A. Giller, L. S. Geita, Z. D. Bleksmit, V. N. Kovalenko, and M. A. Kotovshchikova, “Study of new anticoagulants from a group of indanedione derivatives,” Farmakol. Toksikol., No. 19, 23–27 (1956).

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  3. A. F. Blyuger, S. A. Giller, and B. S. Shenigson, “Detection of anti-lambliasis activity of nitrofurans and first experience with their application for the treatment of human lambliasis invasion,” Med. Parazitol. Parazitar. Bolezni, No. 6, 646–647 (1960).

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  4. É. Ya. Lukevits and S. A. Giller, “Reaction of triethylsilane with mercury salts,” Izv. Akad. Nauk LatvSSR, No. 4, 95–98 (1961).

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  5. É. Ya. Lukevits and S. A. Giller, “[Organosilicon compounds of the furan series.] Syntheses in a series of furan-containing organosilicon compounds. I. Reduction of furyl-, phenyl-, and thienylmercury chlorides with triethylsilane,” Izv. Akad. Nauk LatvSSR, Ser. Khim., 99–102 (1961).

  6. A. I. Meos, L. A. Vol'f, S. A. Giller, S. A. Inkina, and G. P. Sokolov, “Acetalation of polyvinyl alcohol fibers with maleindialdehyde,” Khimicheskie Volokna, 19–21 (1961).

  7. S. A. Giller, L. A. Vol'f, A. I. Meos, and G. P. Sokolov, “Method for waterproofing polyvinyl alcohol fibers,” USSR Author's Certificate No. 138376; Byul. Izobr., No. 10, 44 (1961).

  8. S.A. Giller, G. P. Sokolov, and M. G. Voronkov, “Method for the preparation of alkyl- or aryl-substituted 4-methoxy-2-buten-1-o1,” USSR Author's Certificate No. 162152; Byul. Izobr., No. 9, 26 (1964).

  9. S. A. Giller and Ya. A. Kastron, “Method for the preparation of an epoxide resin,” USSR Author's Certificate No. 167923; Byul. Izobr., No. 3, 38 (1965).

  10. A. A. Avot, M. V. Shimanskaya, and S. A. Giller, “Some problems in the economics of the production of maleic anhydride from furfural,” Izv. Akad. Nauk LatvSSR, No. 10, 87–91 (1965).

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  11. A. S. Shvarts, Ya. A. Kharit, S. A. Giller, K. K. Venter, V. V. Kotetskii, L. A. Vol'f, A. I. Meos, and D. V. Fil'bert, “Method for the preparation of insoles for footwear,” USSR Author's Certificate No. 278468; Byul. Izobr., No. 25, 192 (1970).

  12. B. V. Kurgan, and S. A. Giller, “2-Chlorethylthiol esters of dicarboxylic acids,” Khim. Geterotsikl. Soedin., 12–16 (1970).

  13. A. Ya. Karmil'chik, S. A. Giller, M. V. Shimanskaya, and V. V. Stonkus, “Method for the preparation of benzene,” USSR Author's Certificate No. 266757; Byul. Izobr., No. 32, 207 (1971).

  14. B. V. Kurgan and S. A. Giller, “Opening of the trimethylene sulfide ring,” Khim. Geterotsikl. Soedin., 597–598 (1971).

  15. A. Yu. Tsimanis, N. O. Saldabol, and S. A. Giller, “New method for the synthesis of arylglyoxylic acids,” Zh. Organ. Khim., 8, 2618 (1972).

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  16. S. A. Giller, I. N. Goncharova, Yu. A. Vaintraub, G. S. Gurevich, S. Z. Levin, B. G. Greidin, and V. K. Tsyskovskii, “Method for the preparation of pimelic acid,” USSR Author's Certificate No. 334214; Byul. Izobr., No. 12, 90 (1972).

  17. Z. L. Zosim, L. Ya. Palienko, M. A. Solyanik, N. D. Mikhnovskaya, S. A. Giller, and K. K. Venter, “Method for the modification of cellulose,” USSR Author's Certificate No. 363770; Byul. Izobr., No. 4, 70 (1973).

  18. Ya. Yu. Polis, S. A. Giller, and I. M. Kamyanov, “Method for the preparation of adamantylamino-N-glucuronide,” British Patent No. 1390479 (1975); US Patent No. 3876776 (1975).

Editing

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  9. Khim. Geterotsikl. Soedin. [All-Union Journal], Riga (1965–1975).

  10. Chemistry of Heterocyclic Compounds [in Russian], Vols. 1–3, Zinatne, Riga (1967–1971); Vol. 1, Nitrogen-Containing Heterocycles (1967); Vol. 2, Oxygen-Containing Heterocycles (1970); Vol. 3, Sulfur-Containing Hetrocycles (1971).

  11. Order of the Worker's Red Banner of the Institute of Organic Synthesis, 1957–1969 [in Russian], Zinatne, Riga (1970), second edition (1972).

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  13. “Physiologically and optically active polymeric substances” [Proceedings of the Second All-Union Symposium on the Chemistry and Physical Chemistry of Physiologically and Optically Active Polymeric Substances] [in Russian], Zinatne, Riga (1971).

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  19. Index of Research of the Order of the Worker's Red Banner of the Institute of Organic Synthesis of the Academy of Sciences of the Latvian SSR [in Russian], Liesma, Riga (1974).

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In memory of Solomon Aronovich Giller. Chem Heterocycl Compd 12, 1–26 (1976). https://doi.org/10.1007/BF00473907

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