Abstract
Acetylation and nitrosation of 2,4-diaryl-2-methyl-2,3-dihydro-1H-1,5-benzodiazepines take place at the azomethyne nitrogen. Reduction is stereoselective.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 8, pp. 1122–1126, August, 1987
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Orlov, V.D., Desenko, S.M. & Pivnenko, N.S. Chemical properties of 2,2,4-trisubstituted 2,3-dihydro-1H-1,5-benzodiazepines. Chem Heterocycl Compd 23, 899–902 (1987). https://doi.org/10.1007/BF00473470
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DOI: https://doi.org/10.1007/BF00473470