Skip to main content
SpringerLink
Log in

6-Aminopyrimidine 1-oxides. Acylation and methylation

  • Published:
Chemistry of Heterocyclic Compounds Aims and scope

Abstract

Acylation of 6-aminopyrimidine 1-oxides gives both O- and N-acylation products, but with methylating agents only O-alkyl derivatives are obtained.

This is a preview of subscription content, log in via an institution to check access.

Access this article

Log in via an institution

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Institutional subscriptions

Similar content being viewed by others

Literature Cited

  1. G. Rey-Bellet, R. Reiner, and D. E. Schwartz, Ger. Offen 2,026,997; Chem. Abstr., 74, 76443 (1971).

    Google Scholar 

  2. J. C. Muller and R. Ramuz, Ger. Offen 2,804,518; Chem. Abstr., 89, 197,595 (1978).

    Google Scholar 

  3. T. J. Delia and D. L. Venton, J. Heterocycl. Chem., 9, 73 (1972).

    Google Scholar 

  4. J. M. McCall, R. E. Ten Brink, M. E. Royer, and H. Ko, J. Heterocycl. Chem., 15, 1529 (1978).

    Google Scholar 

  5. V. F. Sedova, T. Yu. Mustafina, and V. P. Mamaev, Khim. Geterotsikl. Soedin., No. 1, 1515 (1981).

    Google Scholar 

  6. R. A. Jones and A. R. Katritzky, J. Chem. Soc., No. 1, 2937 (1960).

    Google Scholar 

  7. L. W. Deady, Synth. Commun., No. 7, 509 (1977).

    Google Scholar 

  8. E. A. Oostveen and H. C. van der Plas, Recl. Trav. Chim., 96, 64 (1977).

    Google Scholar 

  9. S. Takahashi and T. Jatsunami, Chem. Pharm. Bull., 26, 2286 (1978).

    Google Scholar 

  10. R. Peereboom, H. C. van der Plas, and A. Koudius, Recl. Trav. Chim., 93, 58 (1974).

    Google Scholar 

  11. E. Ochiai, Aromatic Amine Oxides, Elsevier, Amsterdam (1967), p. 44.

    Google Scholar 

  12. H. Goncalves, F. Mathis, and C. Foulcher, Bull. Soc. Chim. Fr., No. 7, 2615 (1970).

    Google Scholar 

  13. D. J. Brown and K. Jenega, J. Chem. Soc., Perkin Trans. 1, No. 3, 375 (1974).

    Google Scholar 

  14. D. J. Brown and M. N. Paddon-Row, J. Chem. Soc., C, No. 9, 903 (1967).

    Google Scholar 

  15. N. S. Vostrikov, U. M. Dzhemilev, G. S. Bylina, A. M. Moiseenkov, A. V. Semenovskii, and G. A. Tolstikov, Izv. Akad, Nauk SSSR, Ser. Khim., No. 10, 2337 (1978).

    Google Scholar 

  16. G. S. Bylina, U. M. Dzhemilev, N. S. Vostrikov, G. A. Tolstikov, A. M. Moiseenkov, A. V. Semenovskii, and S. S. Shavanov, Izv. Akad. Nauk SSSR, Ser. Khim., No. 2, 447 (1978).

    Google Scholar 

  17. US Patent No. 3,464,987; Chem. Abstr., 81, 164,337 (1969).

    Google Scholar 

Download references

Author information

Authors and Affiliations

  1. Novosibirsk Branch of the All-Union Scientific Research Institute of Chemical Plant Protectants, 630090, Novosibirsk

    V. F. Sedova & V. P. Mamaev

  2. Novosibirsk Institute of Organic Chemistry, Siberian Branch, Academy of Sciences of the USSR, 630090, Novosibirsk

    V. F. Sedova & V. P. Mamaev

Authors
  1. V. F. Sedova
    View author publications

    You can also search for this author in PubMed Google Scholar

  2. V. P. Mamaev
    View author publications

    You can also search for this author in PubMed Google Scholar

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 11, pp. 1528–1534, November, 1986.

Rights and permissions

Reprints and permissions

About this article

Cite this article

Sedova, V.F., Mamaev, V.P. 6-Aminopyrimidine 1-oxides. Acylation and methylation. Chem Heterocycl Compd 22, 1236–1241 (1986). https://doi.org/10.1007/BF00471809

Download citation

  • Received:

  • Issue Date:

  • DOI: https://doi.org/10.1007/BF00471809

Keywords

Search

Navigation