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Synthesis and biological activity of some thioglycidyl and thietanyl esters of pentavalent phosphorus acids

Conclusions

  1. 1.

    We obtained a number of thioglycidyl and thietanyl esters of pentavalent phosphorus acids.

  2. 2.

    Replacing the thioglycidyl radical by the thietanyl radical in the esters of a dialkoxydithiophosphoric acid leads to the appearance of a well-defined systemic action.

  3. 3.

    The thioglycidyl esters of dialkoxydithio- and dialkoxythiophosphoric acids possess antifungal action toward dermatophytes.

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Literature cited

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    B. A. Arbuzov and O. N. Nuretdinova, Izv. Akad. Nauk SSSR, Ser. Khim., 1314 (1969).

  2. 2.

    O. N. Nuretdinova, F. F. Guseva, and B. A. Arbuzov, Izv. Akad. Nauk SSSR, Ser. Khim., 2851 (1969).

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    O. N. Nuretdinova, Zh. Obshch. Khim.,39, 2141 (1969).

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    W. Lorenz, German Patent No. 1086712 (1961); Ref. Zh., Khim.,19L, 292 (1962).

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    E. Enders and G. Unterstenhofer, US Patent No. 3071594 (1963); Chem. Abstrs.,58, 11330 (1963).

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    K. A. Gar, Methods for Testing the Toxicity and Effectiveness of Insecticides [in Russian], Sel'khozgiz (1963).

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    M. L. Belen'kii, Factors in the Quantitative Evaluation of the Pharmacological Effect [in Russian], Medgiz, Leningrad (1963).

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Additional information

Translated from Izvestiya Akademii Nauk SSSR, Seriya Khimicheskaya, No. 10, pp. 2213–2217, October, 1971.

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Arbuzov, B.A., Nuretdinova, O.N., Neklesova, I.D. et al. Synthesis and biological activity of some thioglycidyl and thietanyl esters of pentavalent phosphorus acids. Russ Chem Bull 20, 2091–2094 (1971). https://doi.org/10.1007/BF00851256

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Keywords

  • Ester
  • Phosphorus
  • Biological Activity
  • Antifungal Action
  • Systemic Action